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MedKoo Chemical Nomenclature
PF-431396 is a potent and selective focal adhesion kinase (FAK) and proline-rich tyrosine kinase 2 (PYK2) inhibitor...
PYR-41 is a ubiquitin-activating enzyme inhibitor (UBE1 inhibitor). PYR-41 blocks ubiquitination reactions but...
CAS#: 2417089-74-6 (S-isomer)
XL177A is a potent USP7 inhibitor. XL177A irreversibly inhibits USP7 with sub-nM potency and selectivity across the...
RG7800, also known as RO6885247 is a potent and selective SMN2 splicing modifier, which is currently under human...
CAS#: 1217457-86-7 (TFA)
GGTI-298 is a potent geranylgeranyltransferase-I (GGTase-I) inhibitor with potential antitumor actrivity. GGTI-298...
CAS#: 957054-30-7 (free base)
Pictilisib, also known as Pictrelisib, GDC-0941, RG7321 and GNE0941 , is an orally bioavailable, and is a potent...
Galeterone, also known as TOK-001 and NX41765; is an orally bioavailable small-molecule androgen receptor modulator...
BAZ2-ICR is an excellent chemical probe for functional studies of the BAZ2 bromodomains in vitro and in vivo. The...
SAG (Smo agonist) free base
CAS#: 912545-86-9 (free base)
SAG is a potent Smoothened (Smo) receptor agonist (Kd = 59 nM); sag antagonizes cyclopamine action at the Smo...
CAS#: 152946-68-4 (HCl salt)
Nolatrexed, also known as AG337, is a thymidylate synthase inhibitor with potential anticancer activity. A phase II...
Retapamulin, also known as SB-275833, is a newer topical agent of pleuromutilin class approved by the Food and Drug...
Flutamide, also known as SCH13521, is a toluidine derivative and nonsteroidal antiandrogen that is structurally...
IKK-16 (free base)
CAS#: 873225-46-8 (free base)
IKK-16 is a potent and slective inhibitor of IκB kinase (IKK) (IC50 values are 40, 70 and 200 nM for IKKβ, IKK...
CAS#: 1428333-96-3 (mseylate)
Pritelivir, also known as AIC-316 and BAY 57-1293, is a potent helicase primase inhibitor. BAY 57-1293 inhibits...
SAN50900, also known as FLT3-IN-3, is a potent and selective FLT3 inhibitor. SAN50900 displays nanomolar activity in...
Elimusertib free base
CAS#: 1876467-74-1 (free base)
Elimusertib, also known as BAY-1895344, is a potent and selective ATM inhibitor. BAY 1895344 shows potent anti-tumor...
Wnt-C59 is a potent porcupine (PORCN) inhibitor. Wnt-C59 inhibits PORCN activity in vitro at nanomolar...
Conoidin A inactivates peroxiredoxins by covalently binding to the catalytic cysteine on the enzyme.
Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.
Aloxistatin (E-64d), is a selective cysteine protease inhibitor or calpain and autophagy inhibitor. E-64d prevents...
CAS#: 1202916-90-2 (free base)
CX-6258 is a pan-Pim kinases inhibitor with excellent biochemical potency and kinase selectivity. CX-6258 exhibited...
C-176 STING inhibitor
C-176 (C-176) is a covalent, in vivo-active, small-molecule inhibitor of STING, attenuates STING-associated...
N-Acetyl calicheamicin is a derivative of calicheamicin, and is a potent enediyne antitumor antibiotic....
Azoramide is a small-molecule modulator of the unfolded protein response with antidiabetic activity. Azoramide...
COH29 is an orally available, aromatically substituted thiazole and inhibitor of the human ribonucleotide reductase...