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PD-123319 free base

CAT#: 555869
CAS#: 130663-39-7 (free base)

PD-123319 is a selective, nonpeptide AT2R antagonist (IC50 = 5.6 nM vs. 100 nM for AT1R). PD-123319 has been used...

SNIPER(CRABP)-11

CAT#: 555560
CAS#: 1384275-50-6

SNIPER(CRABP)-11, also known as PROTAC cIAP1 degrader-4, is a potent protein degrader. SNIPER(CRABP)-11 displayed...

SR-17018

CAT#: 555270
CAS#: 2134602-45-0

SR17018 is an mu-opioid-receptor (MOR) agonist with an EC50 of 97 nM.

Solithromycin

CAT#: 314272
CAS#: 760981-83-7

Solithromycin, also known as CEM-101 and OP-1068, is a ketolide antibiotic undergoing clinical development for the...

Trametinib DMSO solvate

CAT#: 123211
CAS#: 1187431-43-1

Trametinib DMSO solvate is a solvated form of trametinib at 1:1 molar ratio of trametinib to dimethyl sulfoxide....

Amenamevir

CAT#: 319848
CAS#: 841301-32-4

Amenamevir, also known as ASP2151, is a herpes virus helicase-primase inhibitor. ASP2151 had significantly better...

ZK-756326 dihydrochloride

CAT#: 530328
CAS#: 1780259-94-0 (2HCl)

ZK-756326 is a potent, selective and non-peptide CCR8 chemokine receptor agonist. ZK 756326 inhibited the binding of...

PIK-75

CAT#: 202238
CAS#: 372196-67-3 (free base)

PIK-75 was developed as part of a PI 3-kinase drug discovery program. PIK75 attenuates insulin stimulation of Akt/PKB...

Sulfabromomethazine

CAT#: 461673
CAS#: 116-45-0

Sulfabromomethazine, also known as Bromosulfamethazine, NSC 5874, SN 3517, is a long-acting derivative of...

Otenabant HCl

CAT#: 502501
CAS#: 686347-12-6 (HCl)

Otenabant, also known as CP-945,598, is a drug which acts as a potent and highly selective CB1 antagonist. It was...

IKK-16 (free base)

CAT#: 407163
CAS#: 873225-46-8 (free base)

IKK-16 is a potent and slective inhibitor of IκB kinase (IKK) (IC50 values are 40, 70 and 200 nM for IKKβ, IKK...

Olodaterol HCl

CAT#: 329649
CAS#: 869477-96-3 (HCl)

Olodaterol, also known as BI 1744, is a long acting beta-adrenoceptor agonist used as an inhalation for treating...

RXDX-105 (CEP-32496)

CAT#: 205903
CAS#: 1188910-76-0 (free base)

Agerafenib, also known as RXDX-105, CEP-32496 and AC013773, is an orally available v-raf murine sarcoma viral...

UNC2541

CAT#: 407944
CAS#: 1612782-86-1

UNC2541 is a potent and MerTK-specific inhibitor that exhibits sub-micromolar inhibitory activity in the cell-based...

Retapamulin

CAT#: 300270
CAS#: 224452-66-8

Retapamulin, also known as SB-275833, is a newer topical agent of pleuromutilin class approved by the Food and Drug...

SRPIN340

CAT#: 406657
CAS#: 218156-96-8

SRPIN340 is a selective serine arginine protein kinase (SRPK) 1 inhibitor with Ki = 0.89 μM. SRPK1 is a common...

BCH001

CAT#: 463709
CAS#: 384859-58-9

BCH001 is a specific PAPD5 inhibitor that restored telomerase activity and telomere length in DC patient induced...

Diflapolin

CAT#: 471026
CAS#: 724453-98-9

Diflapolin is a potent dual soluble epoxide hydrolase (sEH)/5-lipoxygenase-activating protein (FLAP) inhibitor. It...

Golgicide A

CAT#: 555903
CAS#: 1139889-93-2

Golgicide A is a Potent, selective and reversible inhibitor of GBF1 ArfGEF. Golgicide A inhibited HSV-1 entry via...

Sacubitril calcium salt

CAT#: 314262
CAS#: 1369773-39-6 (hemi-calcium)

Sacubitril, also known as AHU377, is angiotensin receptor neprilysin inhibitor being studied for use in combination...

CX-6258

CAT#: 406247
CAS#: 1202916-90-2 (free base)

CX-6258 is a pan-Pim kinases inhibitor with excellent biochemical potency and kinase selectivity. CX-6258 exhibited...

Entrectinib

CAT#: 206181
CAS#: 1108743-60-7

Entrectinib, also known as RXDX-101 and NMS-E628, is an oral small molecule inhibitor of TrkA, TrkB and TrkC, as well...

Ciproxifan maleate

CAT#: 326719
CAS#: 184025-19-2 (maleate)

Ciproxifan, also known as FUB-359, is an extremely potent histamine H3 inverse agonist/antagonist. Ciproxifan...

PLX5622 fumarate

CAT#: 555654
CAS#: PLX5622 fumarate

PLX5562 is a highly selective brain-penetrant CSF1R inhibitor. In the 5xFAD mouse model of AD, plaques fail to form...

AC-90179 HCl

CAT#: 531399
CAS#: 359878-19-6 (HCl)

AC-90179 is a high selective 5-hydroxytryptamine2A receptor inverse agonist. It is an atypical antipsychotic...