Newest Products

WWL-154

CAT#: 555958
CAS#: 1338574-93-8

WWL-154 is a serine hydrolase inhibitor. Serine hydrolases (SHs) are-one of the largest and most diverse enzyme...

RXDX-105 (CEP-32496)

CAT#: 205903
CAS#: 1188910-76-0 (free base)

Agerafenib, also known as RXDX-105, CEP-32496 and AC013773, is an orally available v-raf murine sarcoma viral...

BI-135585

CAT#: 530402
CAS#: 1114561-85-1

BI-135585 is a potent and selective 11β-HSD1 inhibitor. BI 135585 was safe and well tolerated over 14 days and can be...

NE 52-QQ57

CAT#: 555805
CAS#: 1401728-56-0

NE52-QQ57 is an orally available GPR4 antagonist with an IC50 of 70 nM. NE 52-QQ57 significantly inhibited the...

A286982

CAT#: 531346
CAS#: 280749-17-9

A286982 is an inhibitor that blocks the integrin-ligand interaction between leukocyte function-associated antigen-1...

Seralutinib

CAT#: 585438
CAS#: 1619931-27-9

Seralutinibm, also known as PK-10571 and GB002, is a Novel Inhaled Pdgfr Kinase Inhibitor. Seralutinib demonstrates...

NVS-PAK1-1

CAT#: 561311
CAS#: 1783816-74-9

NVS-PAK1-1 is a specific allosteric PAK1 inhibitor.

DS-1205B

CAT#: 207020
CAS#: 1855860-24-0 (free base)

DS-1205, also known as DS-1205b, is a selective and potent AXL kinase inhibitor with IC50 of 1.3 nM. DS-1205...

HBX19818

CAT#: 562449
CAS#: 1426944-49-1

HBX19818 is a selective inhibitor of USP7.

Conoidin A

CAT#: 555967
CAS#: 18080-67-6

Conoidin A inactivates peroxiredoxins by covalently binding to the catalytic cysteine on the enzyme.

ERD-308

CAT#: 407957
CAS#: 2320561-35-9

ERD-308 is a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Estrogen Receptor (ER) ERD-308 achieves...

BDTX-189

CAT#: 207150
CAS#: 2414572-47-5

BDTX-189 is an orally bioavailable, irreversible, selective, small-molecule inhibitor of certain oncogenic driver,...

BI-894999

CAT#: 206845
CAS#: 1660117-38-3

BI-894999 is a potent and selective BET inhibitor potentially useful for the Treatment of hematological malignancies...

Pyrimorph

CAT#: 561001
CAS#: 868390-90-3

Pyrimorph is a fungicide with high activity against the plant pathogen Phytophthora capsici. Pyrimorph inhibited...

AA41612

CAT#: 574543
CAS#: 433690-62-1

AA41612 is a novel antagonist of melanopsin-mediated phototransduction.

KLH45

CAT#: 562277
CAS#: 1632236-44-2

KLH45 is a selective inhibitor of DDHD2 (DDHD domain containing 2).

WWL229

CAT#: 563210
CAS#: 1338575-28-2

WWL229 is a selective Ces3 inhibitor. It acts by inhibiting recombinant Ces3 but not Ces1f, ABHD6 or other tested...

AQX-016A

CAT#: 555966
CAS#: 849669-54-1

AQX-016A, also known as NSC-741764, is a potent activator of SHIP-1.

ERDRP-0519

CAT#: 563029
CAS#: 1374006-96-8

ERDRP-0519 is an orally available polymerase inhibitor. It shows efficacy against a lethal morbillivirus infection in...

NCGC00262650

CAT#: 574807
CAS#: 344359-25-7

NCGC00262650 is an inhibitor of AMA1-RON2 interaction and c-Src tyrosine kinase activity.

TMP778

CAT#: 522368
CAS#: 1422053-04-0

TMP778 is a novel, potent, and selective RORıt inverse agonist. TMP778 acts potently and selectively to block mouse...

R243

CAT#: 563044
CAS#: 688352-84-3

R243 is an inhibitor of CCR8 signaling and chemotaxis.

BMS-986188

CAT#: 527096
CAS#: 1776115-10-6

BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.

BMS-986187

CAT#: 527097
CAS#: 684238-37-7

BMS-986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.

ML266

CAT#: 555965
CAS#: 1462267-08-8

ML266, also known as CID-4694321, is activator of glucocerebrosidase (GCase). ML266 can serve as starting points to...