MedKoo Biosciences, Inc.
About MedKoo Products
Careers at MedKoo
Remove your patented product from our web
Browse all products
Browse products by research area
Newest stocked products
Frequently asked questions
Process Research & Development
Antibody Drug Conjugation
Hapten Design and Synthesis
How To Order
Terms and Conditions
Download MedKoo Catalogues
Amino Acid Nomenclature Guide
Useful Free Databases
NMR Chemical Shifts of Impurities Charts
MedKoo Chemical Nomenclature
Elemental Period Table
AZD8186 is and inhibitor of the beta isoform of phosphoinositide-3 kinase (PI3K), with potential antineoplastic...
GSK-J4 free base
CAS#: 1373423-53-0 (free base)
GSK-J4 is a cell permeable, potent and selective histone demethylase. GSK-J4 is a prodrug of GSK J1, which is the...
SBE-13 is a selective inhibitor of PLK1 (IC50 values are 200 pM, 875 nM and 66 μ M for PLK1, PLK3 and PLK2...
GSK-461364 is a Polo-like kinase 1 inhibitor, is also a small molecule Polo-like kinase 1 (PLK1) inhibitor with...
GSK-2033 is a potent cell-active LXR antagonist (pIC50 = 7.5). It enhances T-cell proliferation and blocks T...
GSK-189254 free base
CAS#: 720690-73-3 (free base)
GSK-189254 is a potent and selective H3-receptor inverse agonist. It has subnanomolar affinity for the H3 receptor...
Ulodesine, also known as BCX4208, is a purine nucleoside phosphorylase (PNP) inhibitor in development as a once-daily...
CAS#: 686347-12-6 (HCl)
Otenabant, also known as CP-945,598, is a drug which acts as a potent and highly selective CB1 antagonist. It was...
GO 6976, also known as PD-406976, is a potent inhibitor of neurotrophin-receptor intrinsic tyrosine kinase. GÃ¶ 6976...
GNE-477 is a dual inhibitor of PI3K (IC50 = 4 nM for PI3Kα) and mTOR (apparent Ki = 21 nM).
CAS#: 2319647-76-0 (HCl)
OTS514 is a potent TOPK (T-LAK cell-originated protein kinase) inhibitor. OTS514 exhibits growth suppressive effect...
SAR-405 is a potent and selective PIK3C3/Vps34 inhibitor that prevents autophagy and synergizes with MTOR inhibition...
CAS#: 199657-29-9 (HCl)
Givinostat or gavinostat, aslo known as ITF2357, is a potent and orally active histone deacetylase inhibitor with...
CAS#: 69762-85-2 (HCl)
W-9 is a Calmodulin antagonist
CAIX Inhibitor S4
CAIX Inhibitor S4 is an inhibitor of carbonic anhydrase IX. It is selective for CAIX over CAI and CAII but does...
RS 100329 HCl
CAS#: 215654-26-4 (HCl)
RS 100329 is a subtype-selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors). RS 100329...
LYS-006 is a Leukotriene A4 hydrolase (LTA4H) inhibitor for the treatment of Hidradenitis Suppurativa.
NB-360 free base
CAS#: 1262857-73-7 (free base)
NB-360 is a potent and brain penetrable BACE-1 inhibitor. NB-360 shows a superior pharmacological profile and robust...
TCS 2210 is a small molecule inducer of neuronal differentiation.
TCS PIM-1 1
TCS PIM-1 1 is an ATP-competitive Pim-1 kinase inhibitor.
BMS303141 is a potent inhibitor of ATP citrate lyase (ACL). BMS-303141 inhibits lipid synthesis in HepG2 cells with...
CAS#: 1597403-47-8 (trans-isomer)
trans-ISRIB is an Integrated Stress Response Inhibitor. trans-ISRIB inhibits the eIF2α phosphorylation-mediated...
XEN445 is potent and selective endothelial lipase inhibitor, that showed good ADME and PK properties, and...
VU0364439 is a positive allosteric modulator (PAM) of mGlu4 receptors (EC50 = 19.8 nM in vitro for human mGlu4).
ZCL-278 is a cell-permeable inhibitor of Cdc42, a Rho family GTPase.