Newest Products

Ro0711401

CAT#: 532549
CAS#: 714971-87-6

Ro0711401 is a mGlu1 receptor agonist.

PF-573228

CAT#: 406126
CAS#: 869288-64-2

PF-573228 is a potent and selective inhibitor of focal adhesion kinase (FAK) (IC50= 4 nM). Displays 50 - 250-fold...

K-858

CAT#: 407309
CAS#: 72926-24-0

K-858 is a novel inhibitor of mitotic kinesin Eg5 and antitumor agent, induces cell death in cancer cells. K858...

GDC-0077

CAT#: 206818
CAS#: 2060571-02-8

Inavolisib, also known as GDC-0077, is a potent and selective PI3K inhibitor. GDC-0077 blocks an enzyme involved in...

JZL184

CAT#: 510320
CAS#: 1101854-58-3

JZL184 is highly selective, and potent MAGL inhibitor ( monoacylglycerol lipase inhibitor). JZL184 improves behavior...

Gloxazone

CAT#: 558188
CAS#: 2507-91-7

Gloxazone is an effective but toxic anaplasmacide.

Moracin M

CAT#: 556165
CAS#: 56317-21-6

Moracin M is a phosphodiesterase-4 inhibitor isolated from Morus alba. Moracin M has anti-inflammatory activity....

TGP-377421

CAT#: 556164
CAS#: 16752-89-9

TGP-377421, also known as TGP-377/421 and Targapre-miR-377/421, is a potent miR-377 and miR-421 inhibitor that binds...

FEMA-4809

CAT#: 561828
CAS#: 1374760-95-8

FEMA-4809 is a highly potent TRPM8 agonist that is used as a cooling agent.

ZINC30303842

CAT#: 555910
CAS#: 1210906-48-1

ZINC30303842 is a NSD2-PWWP1 antagonist,

Velufenacin

CAT#: 585444
CAS#: 1648737-78-3

Velufenacin is a muscarinic receptor antagonist.

CT52923

CAT#: 556162
CAS#: 205256-55-9

CT52923, also known as KN734, is a platelet-derived growth factor receptor (PDGFR) inhibitor. CT52923 exhibited...

SR18662

CAT#: 408168
CAS#: 2505001-62-5

SR18662 is an optimized anticancel agent based on ML264. SR18662 Efficiently Inhibits the Growth of Colorectal...

MMRi62

CAT#: 408189
CAS#: 352693-80-2

MMRi62 is an MDM4-degrader and apoptosis inducer in leukemia cells. MMRi62 targets MDM4 for degradation and induces...

DXD

CAT#: 207107
CAS#: 1599440-33-1

DXD is an Exatecan derivative and topoisomerase I inhibitor. DXD can be used to make antibody drug conjugate such as...

BMS193885 free base

CAT#: 524448
CAS#: 186185-03-5 (free base)

BMS-193885 is a potent, competitive neuropeptide (NPY) Y1 antagonist (Ki = 3.3 nM, IC50 = 5.9 nM) that displays > 47,...

DWN63831

CAT#: 555968
CAS#: 2409963-83-1

DWN63831 is a lysyl oxidase inhbitor. DWN63831 may be useful in treatment of a variety of disorders, e.g., fibrosis,...

MC-DM1

CAT#: 408188
CAS#: 1375089-56-7

MC-DM is a Maytansine derative and a DM1 molecule with an reactive linker MC. MC-DM1 is a useful precursor to make...

DTP3 inhibitor

CAT#: 555974
CAS#: 1809784-29-9

DTP3 is a selective GADD45β/MKK7 inhibitor, which inhibits cancer-selective NF-κB survival pathway. DTP3 specifically...

SR-18292

CAT#: 530568
CAS#: 2095432-55-4

SR-18292 is a PGC-1α inhibitor. SR-18292 reduces blood glucose, strongly increases hepatic insulin sensitivity, and...

DTHIB

CAT#: 555912
CAS#: 897326-30-6

DTHIB is a direct and selective heat shock factor 1 (HSF1) inhibitor with a Kd of 160 nM. DTHIB physically engages...

ACBI1

CAT#: 556161
CAS#: 2375564-55-7 (free base)

ACBI1 is a potent and cooperative degrader of SMARCA2, SMARCA4 and PBRM1. ACBI1 induced anti-proliferative effects...

Antrodin A

CAT#: 555859
CAS#: 656830-24-9

Antrodin A, also known as AdA and Camphorataanhydride A, is one of the main active ingredients in the solid-state...

Rimiducid

CAT#: 205899
CAS#: 195514-63-7

Rimiducid, also known as AP1903, is a lipid-permeable bivalent "dimerizer" drug that binds FKBP and induces Fas...

VB124

CAT#: 465329
CAS#: 2230186-18-0

VB124 is a novel, highly potent MCT4 inhibitor that mitigated hypertrophy in cultured cardiomyocytes and in mice.