Newest Products

Vaneprim

CAT#: 577816
CAS#: 81523-49-1

Vaneprim is an antibacterial agent.

GNF2133 HCl

CAT#: 555725
CAS#: 2561414-57-9 (HCl)

GNF2133 is a potent and selective DYRK1A inhibitor (IC50 = 6 nM). In vitro, GNF2133 is able to proliferate both...

Icenticaftor

CAT#: 558962
CAS#: 1334546-77-8

Icenticaftor, also known as QBW251 is a Cystic Fibrosis Transmembrane Conductance Regulator Potentiator with Clinical...

GLPG2938

CAT#: 556021
CAS#: 2130996-00-6

GLPG2938 is an antagonists of sphingosine-1-phosphate (S1P) receptor for prophylaxis and/or treatment of diseases...

MM-102 TFA

CAT#: 555880
CAS#: 1883545-52-5 (TFA)

MM-102 is a Potent WDR5/MLL interaction inhibitor. The MM-102 compound prevents the interaction between mixed lineage...

MLS1547

CAT#: 530549
CAS#: 315698-36-3

MLS1547 is a highly efficacious D2 dopamine receptor (D2R) G protein-biased agonist that does not recruit β-arrestin,...

BAY-8400

CAT#: 465423
CAS#: unknown

BAY-8400 is a novel selective inhibitor of DNA-PK. In in vitro studies, BAY-8400 showed synergistic activity of...

MLN120B HCl

CAT#: 532254
CAS#: 1782573-78-7 (2HCl)

MLN-120B is a potent and effective inhibitor of IκB kinase beta subunit (IKKβ) with IC50 value of 20 μM. MLN-120B...

ML-7 HCl

CAT#: 530537
CAS#: 110448-33-4

ML-7 is a MLCK inhibitor. ML-7 inhibits smooth muscle myosin light chain kinase (MLCK) with a Ki value of 0.3 µM....

BIT225

CAT#: 526920
CAS#: 917909-71-8

BIT-225 is a NCp7 zinc finger inhibitor potentially for the treatment of HCV infection and HIV infection. BIT225...

ML364

CAT#: 407457
CAS#: 1991986-30-1

ML364 is a small molecule inhibitor of the deubiquitinase USP2 with potential anticancer activity. ML364 has an IC50...

Eliapixant

CAT#: 574268
CAS#: 1948229-21-7

Eliapixant, also known as BAY 1817080, is a P2X3 receptor antagonist. Eliapixant is both highly potent and selective...

CYM51010

CAT#: 555940
CAS#: 1069498-96-9

CYM51010, also known as CID23723457 and ML335, is a biased ligand of μ-opioid receptor – δ-opioid receptor...

MRTX1719

CAT#: 465753
CAS#: 2630904-45-7

MRTX1719 is a potent and selective binder to the PRMT5•MTA complex and selectively inhibits PRMT5 activity in...

ML329

CAT#: 555752
CAS#: 19992-50-8

ML-329 is an inhibitor of the microphthalmia-associated transcription factor (MITF) pathway with an IC50 value of 1.2...

ML-324

CAT#: 526895
CAS#: 1222800-79-4

ML-324, also known as CID-44143209, is a potent JMJD2 demethylase inhibitor with demonstrated antiviral...

ML311

CAT#: 407459
CAS#: 315698-17-0

ML311, also known as EU-5346, is a potent and selective inhibitor of the Protein-Protein Interaction of Mcl-1 and...

ML277

CAT#: 555789
CAS#: 1401242-74-7

ML277 is a potent activator of KCNQ1 (Kv7.1) channels with >100-fold selectivity versus KCNQ2 and KCNQ4 and no...

ML266

CAT#: 555965
CAS#: 1462267-08-8

ML266, also known as CID-4694321, is activator of glucocerebrosidase (GCase). ML266 can serve as starting points to...

ML-254

CAT#: 555938
CAS#: 1428630-86-7

ML-254, also known as VU0430644; is Positive Allosteric Modulators (PAMs) of mGlu5 with Competitive MPEP-Site...

ML239

CAT#: 408083
CAS#: 1378872-36-6

ML239 is a potent and selective inhibitor of breast cancer stem cells. ML239 was best-in-class with an IC(50)= 1.18...

Rilzabrutinib

CAT#: 462574
CAS#: 1575596-29-0

Rilzabrutinib, also known as PRN1008, is a reversible covalent, selective and oral active inhibitor of Bruton’s...

ML204 HCl

CAT#: 555185
CAS#: 2070015-10-8 (HCl)

ML204 is a novel and potential TRPC4 Channel inhibitor. ML204 inhibited TRPC4β-mediated intracellular Ca(2+) rise...

ML-193

CAT#: 555262
CAS#: 713121-80-3

ML-193, also known as CID 1261822, is a potent antagonist of GPR55 (IC50 = 221 nM).

ML192

CAT#: 522625
CAS#: 460331-61-7

ML192, also known as MLS000526305 and CID1434953, is a selective ligands for GPR55. The orphan G protein coupled...