Metiprenaline HCl

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 125350

CAS#: 1420-27-5 (HCl)

Description: Metiprenaline was developed as a bronchodilator.

Chemical Structure

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Metiprenaline HCl
CAS# 1420-27-5 (HCl)
Instruction

Theoretical Analysis

MedKoo Cat#: 125350
Name: Metiprenaline HCl
CAS#: 1420-27-5 (HCl)
Chemical Formula: C12H20ClNO3
Exact Mass: 261.11
Molecular Weight: 261.750
Elemental Analysis: C, 55.07; H, 7.70; Cl, 13.54; N, 5.35; O, 18.34

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

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Related CAS #: 1420-27-5 (HCl)  

Synonym: 1420-27-5; alpha-((Isopropylamino)methyl)vanillyl alcohol hydrochloride; 13015-70-8; alpha-[(Isopropylamino)methyl]vanillyl alcohol hydrochloride; EINECS 235-872-3; metiprenaline hydrochloride

IUPAC/Chemical Name: 4-(1-hydroxy-2-(isopropylamino)ethyl)-2-methoxyphenol hydrochloride

InChi Key: FBJGAKKBRRBUOG-UHFFFAOYSA-N

InChi Code: InChI=1S/C12H19NO3.ClH/c1-8(2)13-7-11(15)9-4-5-10(14)12(6-9)16-3;/h4-6,8,11,13-15H,7H2,1-3H3;1H

SMILES Code: Cl.COC1=C(O)C=CC(=C1)C(O)CNC(C)C

Appearance: To be determined

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).

Solubility: To be determined

Shelf Life: >2 years if stored properly

Drug Formulation: To be determined

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 261.75 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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7: Bryan-Lluka LJ, Westwood NN, O'Donnell SR. Vascular uptake of catecholamines in perfused lungs of the rat occurs by the same process as Uptake1 in noradrenergic neurones. Naunyn Schmiedebergs Arch Pharmacol. 1992 Mar;345(3):319-26. PubMed PMID: 1535692.

8: Schömig E, Schönfeld CL. Extraneuronal noradrenaline transport (uptake2) in a human cell line (Caki-1 cells). Naunyn Schmiedebergs Arch Pharmacol. 1990 May;341(5):404-10. PubMed PMID: 2164161.

9: Schömig E, Babin-Ebell J, Schönfeld CL, Russ H, Trendelenburg U. Human Caki-1 cells are the first model for extraneuronal transport of noradrenaline (uptake2) which is based on a clonal cell line. J Neural Transm Suppl. 1990;32:437-40. PubMed PMID: 2089108.

10: Causon RC, Brown MJ, Davies DS. Reversed-phase high-performance liquid chromatography and amperometric detection of 3-O-methyl isoprenaline sulphate: application to studies on the presystemic metabolism of d-isoprenaline in man. J Chromatogr. 1985 Feb 8;337(2):311-20. PubMed PMID: 3988861.