Etilefrine hydrochloride
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MedKoo CAT#: 592558

CAS#: 943-17-9 (HCl)

Description: Etilefrine hydrochloride is an adrenergic agonist that appears to interact with beta-2 and some alpha adrenergic receptors. It has been used as a vasoconstrictor agent.

Chemical Structure

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Etilefrine hydrochloride
CAS# 943-17-9 (HCl)
Instruction

Theoretical Analysis

MedKoo Cat#: 592558
Name: Etilefrine hydrochloride
CAS#: 943-17-9 (HCl)
Chemical Formula: C10H16ClNO2
Exact Mass: 217.09
Molecular Weight: 0.000
Elemental Analysis: C, 55.17; H, 7.41; Cl, 16.28; N, 6.43; O, 14.70

Price and Availability

Size Price Availability Quantity
1g USD 285 2 Weeks
5g USD 585 2 Weeks
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Related CAS #: 943-17-9 (HCl)   709-55-7 (free base)   95670-87-4 (S-isomer HCl)   95670-88-5 (R-isomer HCl)    

Synonym: Etilefrine hydrochloride; Ethyl adrianol

IUPAC/Chemical Name: alpha-((Ethylamino)methyl)-m-hydroxybenzyl alcohol hydrochloride

InChi Key: KTNROWWHOBZQGK-UHFFFAOYSA-N

InChi Code: InChI=1S/C10H15NO2.ClH/c1-2-11-7-10(13)8-4-3-5-9(12)6-8;/h3-6,10-13H,2,7H2,1H3;1H

SMILES Code: OC1=CC(C(O)CNCC)=CC=C1.[H]Cl

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 0.00 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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13: Ohkura Y, Ueno M, Iizuka T, Haruta S, Tanaka T, Udagawa H. New Combined Medical Treatment With Etilefrine and Octreotide for Chylothorax After Esophagectomy: A Case Report and Review of the Literature. Medicine (Baltimore). 2015 Dec;94(49):e2214. doi: 10.1097/MD.0000000000002214. PubMed PMID: 26656358; PubMed Central PMCID: PMC5008503.

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