TM2 TEAD inhibitor
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 125069

CAS#: 1008768-41-9

Description: TM2 TEAD inhibitor is a potent and reversible TEA domain transcription factor inhibitor.

Chemical Structure

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TM2 TEAD inhibitor
CAS# 1008768-41-9
Instruction

Theoretical Analysis

MedKoo Cat#: 125069
Name: TM2 TEAD inhibitor
CAS#: 1008768-41-9
Chemical Formula: C26H33N3O3
Exact Mass: 435.25
Molecular Weight: 435.570
Elemental Analysis: C, 71.70; H, 7.64; N, 9.65; O, 11.02

Price and Availability

Size Price Availability Quantity
10mg USD 350 2 Weeks
50mg USD 1050 2 Weeks
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Synonym: TM2 TEAD inhibitor; TM2 TEAD-inhibitor; TM2-TEAD inhibitor

IUPAC/Chemical Name: 4-(3-(2-cyclohexylethoxy)benzoyl)-N-phenylpiperazine-1-carboxamide

InChi Key: LWLAYULJAJMPKG-UHFFFAOYSA-N

InChi Code: InChI=1S/C26H33N3O3/c30-25(22-10-7-13-24(20-22)32-19-14-21-8-3-1-4-9-21)28-15-17-29(18-16-28)26(31)27-23-11-5-2-6-12-23/h2,5-7,10-13,20-21H,1,3-4,8-9,14-19H2,(H,27,31)

SMILES Code: O=C(N1CCN(CC1)C(C2=CC(OCCC3CCCCC3)=CC=C2)=O)NC4=CC=CC=C4

Appearance: To be determined

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).

Solubility: To be determined

Shelf Life: >2 years if stored properly

Drug Formulation: To be determined

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 435.57 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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