Newest Products

Plitidepsin

CAT#: 200150
CAS#: 137219-37-5

Plitidepsin is a cyclic depsipeptide isolated from the marine tunicate Aplidium albicans. Plitidepsin displays a...

PFK-158

CAT#: 206166
CAS#: 1462249-75-7

PFK-158, also known as ACT-PFK-158, is an inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatases...

GABOB (beta-hydroxy-GABA)

CAT#: 319920
CAS#: 7013-05-0

GABOB, also known as γ-Amino-β-hydroxybutyric acid, β-hydroxy-γ-aminobutyric acid, β-hydroxy-GABA, is an...

HSF1A

CAT#: 555224
CAS#: 1196723-93-9

HSF1A is an activator of Heat shock transcription factor 1 (HSF1).

HS-1793

CAT#: 408136
CAS#: 927885-00-5

HS-1793 is a resveratrol analogue. HS-1793 downregulates the expression of hypoxia-induced HIF-1 and VEGF and...

HMN-154

CAT#: 555217
CAS#: 173528-92-2

HMN-154 is a benzenesulfonamide anticancer agent. HMN-154 inhibits DNA binding of NF-Y to the human major...

Entrectinib

CAT#: 206181
CAS#: 1108743-60-7

Entrectinib, also known as RXDX-101 and NMS-E628, is an oral small molecule inhibitor of TrkA, TrkB and TrkC, as well...

Elimusertib free base

CAT#: 333061
CAS#: 1876467-74-1 (free base)

Elimusertib, also known as BAY-1895344, is a potent and selective ATM inhibitor. BAY 1895344 shows potent anti-tumor...

HBX19818

CAT#: 562449
CAS#: 1426944-49-1

HBX19818 is a selective inhibitor of USP7.

Radotinib

CAT#: 205990
CAS#: 926037-48-1 (free base)

Radotinib, also known as IY-5511, is an orally available, a second-generation tyrosine kinase inhibitor of Bcr-Abl...

GNF-7

CAT#: 407257
CAS#: 839706-07-9

GNF-7 is a type-II T315I inhibitor. GNF-7 inhibits Ack1 and germinal center kinase (GCK). GNF-7 displayed...

H3B-5942 free base

CAT#: 408068
CAS#: 2052128-15-9 (free base)

H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist. In vitro comparisons...

GW806742X

CAT#: 408128
CAS#: 579515-63-2

GW806742X is a potent MLKL inhibitor, also a human and murine necroptosis inhibitor. GW806742X binds the MLKL...

GW284543

CAT#: 555674
CAS#: 790186-68-4

GW284543, also known as UNC10225170;, is a potent and selective MEK5 inhibitor with the potential for cancer...

GW280264X

CAT#: 555806
CAS#: 866924-39-2

GW280264X is an ADAM17 inhibitor.

XL092

CAT#: 555990
CAS#: 2367004-54-2

XL092 is an ATP-competitive inhibitor of multiple RTKs including MET, VEGFR2, AXL and MER, with IC50 values in...

GSK805

CAT#: 555509
CAS#: 1426802-50-7

GSK805, also known as ROR gamma-t-IN-1, is a potent, orally bioavailable retinoid-related orphan receptor gamma t...

GSK6853

CAT#: 406745
CAS#: 1910124-24-1

GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain,...

GSK620

CAT#: 555971
CAS#: 2088410-46-0

GSK620 is a Potent, selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2)...

HM43239

CAT#: 207171
CAS#: 2569527-64-4

HM43239 is an orally active small molecule inhibitor of FLT3 that selectively inhibits not only FLT3 wild type, ITD...

BAY-1251152 racemate

CAT#: 207142
CAS#: 1610358-53-6 (racemate)

BAY-1251152 racemate, also known as (±)-BAY-1251152, is a racemic mixture of BAY-1251152. BAY-1251152 is a potent and...

GSK4112

CAT#: 531875
CAS#: 1216744-19-2

GSK4112 is a selective Rev-Erbα agonist (EC50 = 250 nM). GSK4112 enhances recruitment of nuclear receptor...

GSK3i XIII

CAT#: 562298
CAS#: 404828-08-6

GSK3i XIII is an ATP-binding site inhibitor of GSK-3.

SGI-7079

CAT#: 206483
CAS#: 1239875-86-5

SGI-7079 is a potent and selective Axl inhibitor with potential anticancer activity. SGI-7079 effectively inhibited...

GSK3039294

CAT#: 555377
CAS#: 1819986-22-5

GSK3039294 is an orally available small molecule inhibitor of serum amyloid P component (SAP) binding to amyloid...