AZD-6280
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 524349

CAS#: 942436-93-3

Description: AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder.


Chemical Structure

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AZD-6280
CAS# 942436-93-3

Theoretical Analysis

MedKoo Cat#: 524349
Name: AZD-6280
CAS#: 942436-93-3
Chemical Formula: C20H22N4O3
Exact Mass: 366.17
Molecular Weight: 366.410
Elemental Analysis: C, 65.56; H, 6.05; N, 15.29; O, 13.10

Price and Availability

Size Price Availability Quantity
50mg USD 550
100mg USD 950
200mg USD 1650
500mg USD 2150
1g USD 2950
2g USD 4850
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Synonym: AZD-6280; AZD6280; AZD 6280;

IUPAC/Chemical Name: 3-Cinnolinecarboxamide, 4-amino-8-(2,5-dimethoxyphenyl)-N-propyl-

InChi Key: NVWCZRPXYVDQEE-UHFFFAOYSA-N

InChi Code: InChI=1S/C20H22N4O3/c1-4-10-22-20(25)19-17(21)14-7-5-6-13(18(14)23-24-19)15-11-12(26-2)8-9-16(15)27-3/h5-9,11H,4,10H2,1-3H3,(H2,21,23)(H,22,25)

SMILES Code: CCCNC(=O)c1c(c2cccc(c2nn1)c3cc(ccc3OC)OC)N

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 366.41 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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