WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 466001
CAS#: 536702-12-2
Description: G2iA is a novel potent GLUT2‑selective inhibitor (IC50 of 0.61 µM).
MedKoo Cat#: 466001
Name: G2iA
CAS#: 536702-12-2
Chemical Formula: C27H24FN3O2S
Exact Mass: 473.1573
Molecular Weight: 473.5664
Elemental Analysis: C, 68.48; H, 5.11; F, 4.01; N, 8.87; O, 6.76; S, 6.77
This product is not in stock, which may be available by custom synthesis.
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Synonym: G2iA; G2-iA; G2 iA;
IUPAC/Chemical Name: 1-(5-(4-fluorophenyl)-3-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-1-yl)-2-((2-methyl-1H-indol-3-yl)thio)ethan-1-one
InChi Key: OWPBTSFHLNARSW-UHFFFAOYSA-N
InChi Code: InChI=1S/C27H24FN3O2S/c1-17-27(22-5-3-4-6-23(22)29-17)34-16-26(32)31-25(19-7-11-20(28)12-8-19)15-24(30-31)18-9-13-21(33-2)14-10-18/h3-14,25,29H,15-16H2,1-2H3
SMILES Code: O=C(N1N=C(C2=CC=C(OC)C=C2)CC1C3=CC=C(F)C=C3)CSC4=C(C)NC5=C4C=CC=C5
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: To be determined
Shelf Life: >2 years if stored properly
Drug Formulation: To be determined
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 473.5664 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
