GLPG2938
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 556021

CAS#: 2130996-00-6

Description: GLPG2938 is an antagonists of sphingosine-​1-​phosphate (S1P) receptor for prophylaxis and​/or treatment of diseases including fibrotic, inflammatory, autoimmune, metabolic, cardiovascular, and​/or proliferative diseases. GLPG2938 displayed S1P inhibitory activity.with EC50 value of 9.5 nM (S1P2 antagonist EC50)​.


Chemical Structure

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GLPG2938
CAS# 2130996-00-6

Theoretical Analysis

MedKoo Cat#: 556021
Name: GLPG2938
CAS#: 2130996-00-6
Chemical Formula: C20H19F6N7O2
Exact Mass: 503.1504
Molecular Weight: 503.4094
Elemental Analysis: C, 47.72; H, 3.80; F, 22.64; N, 19.48; O, 6.36

Price and Availability

Size Price Availability Quantity
50.0mg USD 1250.0 2 Weeks
100.0mg USD 1950.0 2 Weeks
200.0mg USD 3250.0 2 Weeks
500.0mg USD 4250.0 2 Weeks
1.0g USD 6950.0 2 Weeks
2.0g USD 8950.0 2 Weeks
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Synonym: MUN96006; MUN-96006; MUN 96006; GLPG2938; GLPG-2938; GLPG 2938;

IUPAC/Chemical Name: 1-(2-ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea

InChi Key: MGJMUVKYINFAQC-UHFFFAOYSA-N

InChi Code: InChI=1S/C20H19F6N7O2/c1-4-35-15-7-11(6-14(29-15)19(21,22)23)28-18(34)27-8-12-5-10(2)16(31-30-12)13-9-33(3)32-17(13)20(24,25)26/h5-7,9H,4,8H2,1-3H3,(H2,27,28,29,34)

SMILES Code: O=C(NCC1=NN=C(C2=CN(C)N=C2C(F)(F)F)C(C)=C1)NC3=CC(OCC)=NC(C(F)(F)F)=C3

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: To be determined

Shelf Life: >2 years if stored properly

Drug Formulation: To be determined

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 503.4094 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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GLPG2938

50.0mg / USD 1250.0