BDZ-g

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 564438

CAS#: 732278-52-3

Description: BDZ-g is a potent inhibitor of both the closed-channel and the open-channel conformations of all four homomeric AMPA receptor channels, as well as two GluA2R containing complex AMPA receptor channels.


Price and Availability

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BDZ-g is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 564438
Name: BDZ-g
CAS#: 732278-52-3
Chemical Formula: C21H21N5O2S
Exact Mass: 407.1416
Molecular Weight: 407.49
Elemental Analysis: C, 61.90; H, 5.19; N, 17.19; O, 7.85; S, 7.87


Synonym: BDZg; BDZ g; BDZ-g; GYKI47409; GYKI-47409; GYKI 47409

IUPAC/Chemical Name: (R)-5-(4-Amino-3-methyl-phenyl)-8-methyl-7-(5-methyl-1,3,4-thiadiazol-2-yl)-8,9-dihydro-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine

InChi Key: DBDUGNPURSLMPS-GFCCVEGCSA-N

InChi Code: InChI=1S/C21H21N5O2S/c1-11-6-14(4-5-17(11)22)20-16-9-19-18(27-10-28-19)8-15(16)7-12(2)26(25-20)21-24-23-13(3)29-21/h4-6,8-9,12H,7,10,22H2,1-3H3/t12-/m1/s1

SMILES Code: CC1=NN=C(N2N=C(C3=CC=C(N)C(C)=C3)C4=CC(OCO5)=C5C=C4C[C@H]2C)S1


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO

Shelf Life:
>3 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
2934.99.03.00