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MedKoo CAT#: 558399

CAS#: 1395048-49-3

Description: M-110 is a inhibitor of protein arginine N-methyltransferases (PRMTs). It is also a highly isoform-selective, cell permeable and potent ATP-competitive inhibitor of the PIM kinase family that prefers PIM-3, shown to inhibit the proliferation of prostate cancer cell lines with IC50s between 0.6 to 0.9 μM, with no activity on normal human peripheral blood mononuclear cells up to 40 μM.

Price and Availability

Size Price Shipping out time Quantity
5mg USD 270 2 Weeks
25mg USD 460 2 Weeks
Inquire bulk and customized quantity

Pricing updated 2020-09-29. Prices are subject to change without notice.

M-110, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 558399
Name: M-110
CAS#: 1395048-49-3
Chemical Formula: C22H28ClN5O3
Exact Mass: 445.19
Molecular Weight: 445.95
Elemental Analysis: C, 59.25; H, 6.33; Cl, 7.95; N, 15.70; O, 10.76

Synonym: M-110; M 110; M110;

IUPAC/Chemical Name: (E)-2-(3-Morpholin-4-yl-propylamino)-isonicotinic acid [1-(4-chloro-2-hydroxy-phenyl)-propylidene]-hydrazide


InChi Code: InChI=1S/C22H28ClN5O3/c1-2-19(18-5-4-17(23)15-20(18)29)26-27-22(30)16-6-8-25-21(14-16)24-7-3-9-28-10-12-31-13-11-28/h4-6,8,14-15,29H,2-3,7,9-13H2,1H3,(H,24,25)(H,27,30)/b26-19+


Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>3 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:


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