WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 563277
CAS#: 862250-23-5
Description: FCPT is an ATP competitive inhibitor of kinesin-5.
MedKoo Cat#: 563277
Name: FCPT
CAS#: 862250-23-5
Chemical Formula: C17H13FN2S
Exact Mass: 296.0783
Molecular Weight: 296.36
Elemental Analysis: C, 68.90; H, 4.42; F, 6.41; N, 9.45; S, 10.82
This product is not in stock, which may be available by custom synthesis.
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Synonym: FCPT;
IUPAC/Chemical Name: 2-(1-(4-Fluorophenyl)cyclopropyl)-4-(pyridin-4-yl)thiazole
InChi Key: PVPYZVCHGWNKFZ-UHFFFAOYSA-N
InChi Code: InChI=1S/C17H13FN2S/c18-14-3-1-13(2-4-14)17(7-8-17)16-20-15(11-21-16)12-5-9-19-10-6-12/h1-6,9-11H,7-8H2
SMILES Code: FC1=CC=C(C2(C3=NC(C4=CC=NC=C4)=CS3)CC2)C=C1
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.03.00
The following data is based on the product molecular weight 296.36 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
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