p38alpha-IN-4

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 562371

CAS#: 1006378-90-0

Description: p38alpha-IN-4 is a reversible p38alpha MAP kinase inhibitor.


Price and Availability

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p38alpha-IN-4 is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 562371
Name: p38alpha-IN-4
CAS#: 1006378-90-0
Chemical Formula: C21H14F2N2O
Exact Mass: 348.1074
Molecular Weight: 348.35
Elemental Analysis: C, 72.41; H, 4.05; F, 10.91; N, 8.04; O, 4.59


Synonym: p38alpha-IN-4; p38alpha IN 4; p38alphaIN4; p38alpha inhibitor 4; p38alpha-inhibitor-4; p38 MAP Kinase Inhibitor XI;

IUPAC/Chemical Name: 4-(2,4-Difluorophenyl)-8-(2-methylphenyl)-1,7-naphthyridine-7-oxide

InChi Key: BSZQSLWNMVTKJT-UHFFFAOYSA-N

InChi Code: InChI=1S/C21H14F2N2O/c1-13-4-2-3-5-15(13)21-20-18(9-11-25(21)26)16(8-10-24-20)17-7-6-14(22)12-19(17)23/h2-12H,1H3

SMILES Code: [O-][N+]1=C(C2=CC=CC=C2C)C3=NC=CC(C4=CC=C(F)C=C4F)=C3C=C1


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
293490


References

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