XU1

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 526596

CAS#: 53439-81-9

Description: XU1 is a potent and selective pan Aurora inhibitor; Phosphorylation of histone H3 (pHH3) inhibitor.


Price and Availability

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Price

Size
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Size
Price

XU1 is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 526596
Name: XU1
CAS#: 53439-81-9
Chemical Formula: C12H8N2O
Exact Mass: 196.0637
Molecular Weight: 196.209
Elemental Analysis: C, 73.46; H, 4.11; N, 14.28; O, 8.15


Synonym: XU1

IUPAC/Chemical Name: 5H-Benzo[c][1,8]naphthyridin -6-one

InChi Key: YLSBDRGLLZDAKB-UHFFFAOYSA-N

InChi Code: InChI=1S/C12H8N2O/c15-12-10-5-2-1-4-8(10)9-6-3-7-13-11(9)14-12/h1-7H,(H,13,14,15)

SMILES Code: O=C1NC2=NC=CC=C2C3=CC=CC=C13


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
293490


References

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D, He J, Chen H, Jin L, Rota PA, Xu W. Epidemiologic and genetic characteristics
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19: Xu K, Butlin M, Avolio AP. Effects of pressure-dependent segmental arterial
compliance and postural changes on pulse wave transmission in an arterial model
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