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MedKoo CAT#: 571274

CAS#: 65372-80-7

Description: AA560 is a nonsteroidal antiandrogen. AA560 decreases the uptake of 3H-androgens in the ventral prostate. AA560 decreases the weight of accessory organs.

Price and Availability

Size Price Shipping out time Quantity
Inquire bulk and customized quantity

Pricing updated 2020-03-29. Prices are subject to change without notice.

AA560 is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 571274
Name: AA560
CAS#: 65372-80-7
Chemical Formula: C10H10Cl3NO2
Exact Mass: 280.9777
Molecular Weight: 282.55
Elemental Analysis: C, 42.51; H, 3.57; Cl, 37.64; N, 4.96; O, 11.32

Synonym: AA560; AA-560; AA 560

IUPAC/Chemical Name: Propanamide, 2-hydroxy-2-methyl-N-(3,4,5-trichlorophenyl)-


InChi Code: InChI=1S/C10H10Cl3NO2/c1-10(2,16)9(15)14-5-3-6(11)8(13)7(12)4-5/h3-4,16H,1-2H3,(H,14,15)

SMILES Code: CC(C)(O)C(NC1=CC(Cl)=C(Cl)C(Cl)=C1)=O

Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:


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2: Yoshida M, Asano M, Kaetsu I, Yamanaka H, Nakai K, Yuasa H, Shida K. Effect of drug-vinyl copolymer delivery composites on the rat prostate. J Biomed Mater Res. 1985 Jul-Aug;19(6):615-29. PubMed PMID: 2416759.

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11: Yamanaka H, Matsuoka M, Yuasa H, Koya A, Imai K, Ebihara K, Nakai K, Shida K. Effects of antiprostatic agents on 5alpha-dihydrotestosterone binding to rat hypophyseal and hypothalamic cytosol macromolecules. Endocrinol Jpn. 1979 Feb;26(1):97-102. PubMed PMID: 86441.

12: Benvenga S, Bartolone L, Trimarchi F. Thyroid iodide transporter: local sequence homologies with thyroid autoantigens. J Endocrinol Invest. 1997 Oct;20(9):508-12. PubMed PMID: 9413803.

13: Suzuki T, Horibe I, Uchida N, Ezumi K, Uchida K, Takeda K, Tanaka A, Nishizawa Y, Matsumoto K. Effects of antiandrogens on growth of androgen-dependent mouse mammary tumor (Shionogi carcinoma 115) in vivo and in vitro. J Steroid Biochem Mol Biol. 1990 Nov 30;37(4):559-67. PubMed PMID: 2278840.