Acetildenafil
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 561226

CAS#: 831217-01-7

Description: Acetildenafil is a synthetic drug which acts as a phosphodiesterase inhibitor. It is an analog of sildenafil (Viagra) which has been detected in numerous different brands of supposedly "herbal" aphrodisiac products sold to boost libido and alleviate erectile dysfunction.


Chemical Structure

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Acetildenafil
CAS# 831217-01-7

Theoretical Analysis

MedKoo Cat#: 561226
Name: Acetildenafil
CAS#: 831217-01-7
Chemical Formula: C25H34N6O3
Exact Mass: 466.2692
Molecular Weight: 466.59
Elemental Analysis: C, 64.36; H, 7.35; N, 18.01; O, 10.29

Price and Availability

Size Price Availability Quantity
1.0mg USD 235.0 2 Weeks
5.0mg USD 540.0 2 Weeks
10.0mg USD 900.0 2 Weeks
25.0mg USD 1565.0 2 Weeks
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Synonym: Acetildenafil; Hongdenafil

IUPAC/Chemical Name: 5-[2-Ethoxy-5-[2-(4-ethylpiperazin-1-yl)acetyl]phenyl]-1-methyl-3-propyl-4H-pyrazolo[4,3-d]pyrimidin-7-one

InChi Key: RRBRQNALHKQCAI-UHFFFAOYSA-N

InChi Code: InChI=1S/C25H34N6O3/c1-5-8-19-22-23(29(4)28-19)25(33)27-24(26-22)18-15-17(9-10-21(18)34-7-3)20(32)16-31-13-11-30(6-2)12-14-31/h9-10,15H,5-8,11-14,16H2,1-4H3,(H,26,27,33)

SMILES Code: O=C1C(N(C)N=C2CCC)=C2NC(C3=CC(C(CN4CCN(CC)CC4)=O)=CC=C3OCC)=N1

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 466.59 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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