Gavestinel Sodium

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MedKoo CAT#: 529421

CAS#: 153436-38-5 (sodium)

Description: Gavestinel Sodium is an NMDA glycine-site antagonist potentially for the treatment of stroke.

Price and Availability

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Pricing updated 2020-03-29. Prices are subject to change without notice.

Gavestinel Sodium is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to to inquire quote.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 529421
Name: Gavestinel Sodium
CAS#: 153436-38-5 (sodium)
Chemical Formula: C18H11Cl2N2NaO3
Exact Mass:
Molecular Weight: 397.18
Elemental Analysis: C, 54.43; H, 2.79; Cl, 17.85; N, 7.05; Na, 5.79; O, 12.08

Related CAS #: 153436-22-7 (free base)   153436-38-5 (sodium)  

Synonym: GV-150526A; GV150526A; GV 150526A

IUPAC/Chemical Name: sodium (E)-4,6-dichloro-3-(3-oxo-3-(phenylamino)prop-1-en-1-yl)-1H-indole-2-carboxylate


InChi Code: InChI=1S/C18H12Cl2N2O3.Na/c19-10-8-13(20)16-12(17(18(24)25)22-14(16)9-10)6-7-15(23)21-11-4-2-1-3-5-11;/h1-9,22H,(H,21,23)(H,24,25);/q;+1/p-1/b7-6+;

SMILES Code: O=C(C(N1)=C(/C=C/C(NC2=CC=CC=C2)=O)C3=C1C=C(Cl)C=C3Cl)[O-].[Na+]

Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:


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