Gaboxadol HCl

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MedKoo CAT#: 525150

CAS#: 85118-33-8 (HCl)

Description: Gaboxadol, also known as THIP, OV-101; Lu-02-030; MK-0928; Lu-02030, is a GABA agonist. It is an inhibitor of GABA uptake systems. Gaboxadol can also be a non-opioid analgesic and a novel type of hypnotic.

Price and Availability

Size Price Shipping out time Quantity
25mg USD 150 2 Weeks
50mg USD 250 2 Weeks
100mg USD 450 2 Weeks
200mg USD 850 2 Weeks
500mg USD 1750 2 Weeks
1g USD 2950 2 Weeks
2g USD 4950 2 Weeks
5g USD 7950 2 Weeks
Inquire bulk and customized quantity

Pricing updated 2020-06-02. Prices are subject to change without notice.

Gaboxadol HCl, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 525150
Name: Gaboxadol HCl
CAS#: 85118-33-8 (HCl)
Chemical Formula: C6H9ClN2O2
Exact Mass: 140.05858
Molecular Weight: 176.6
Elemental Analysis: C, 40.81; H, 5.14; Cl, 20.07; N, 15.86; O, 18.12

Synonym: Gaboxadol; OV-101; Lu-02-030; MK-0928; Lu-02030; OV-101; Lu02-030; MK0928; Lu02030. THIP

IUPAC/Chemical Name: 4,5,6,7-Tetrahydroisoxazolo(5,4-c)pyridin-3(2H)-one monohydrochloride


InChi Code: InChI=1S/C6H8N2O2.ClH/c9-6-4-1-2-7-3-5(4)10-8-6;/h7H,1-3H2,(H,8,9);1H


Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:

Additional Information

Related CAS#
CAS#64603-91-4 (Gaboxadol freebase)
CAS#85118-33-8 (Gaboxadol hydrochloride salt)
CAS#65202-63-3 (Gaboxadol hydrobromide salt)


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