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MedKoo's Collection:

New anticancer agents under worldwide clinical trials

(last update: Feb 13, 2013)

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Cat#      ||  Product name

201830  ||  2-methoxyestradiol (angiogenesis inhibitor)

200880  ||  4-demethylpenclomedine(DMPEN) (alkylation agent)

205800  ||  4SC-202 (HDAC inhibitor)

205802  ||  4SC-203 (multi-target kinase inhibitor)

205804  ||  4SC-205 (human kinesin spindle protein Eg5 inhibitor)

202170  ||  Abexinostat(PCI-24781;  CRA-024781) (HDAC inhibitor)

205806  ||  ABC294640 (sphingosine kinase-2 inhibitor)

100011  ||  Abiraterone (androgen biosynthesis inhibitor)

200030  ||  Abiraterone acetate (androgen biosynthesis inhibitor)

202852  ||  ABR-215050 (Tasquinimod) (angiogenic inhibitor)

205807  ||  ABT-199 (BCL inhibitor)

201970  ||  ABT-263 (Novitoclax) (Bcl-2 Inhibitor)

204140  ||  ABT-348 (receptor tyrosine kinase inhibitor)

206044  ||  ABT-414 (EGFR inhibitor)

205761  ||  ABT-510 (angiogenesis inhibitor)

200040  ||  ABT-518 (MMP inhibitor)

205896  ||  ABT-700 (c-MET inhibitor)

200044  ||  ABT-737 (BCL-2 inhibitor)

200050  ||  ABT-751 (Microtubule Inhibitor)

205762  ||  ABT-767 (PARP inhibitor)

205897  ||  AC430 (JAK2 inhibitor)

200078  ||  AC480 (BMS-599626) (HER inhibitor)

200079  ||  Acadesine (AMP-activated protein kinase activator)

204170  ||  Acolbifene (selective estrogen receptor modulator)

205808  ||  ACY-1215 (HDAC6 inhibitor)

201823  ||  Acyline (MER-104) (GnRH antagonist)

204180  ||  AD-1001 (immunomodulatory therapy)

200080  ||  Aderbasib (INCB007839) (sheddase inhibitor)

200090  ||  ADPM06 (PDT photosensitizer)

202042  ||  ADW742 (NVP-ADW742) (IGF-IR inhibitor)

200100  ||  AEE788 (EGFR, ErbB2, KDR, and Flt-1 inhibitor)

201475  ||  AEG-40826 (HGS-1029) (IAP Inhibitor)

200110  ||  AEG-41174 ( tyrosine kinase inhibitor)

204210  ||  AEW-541 (NVP-AEW541) (IGF-IR inhibitor)

204220  ||  AEZS-108 (AN-152) (LHRH-receptor specified doxorubicin conjugate)

200115  ||  AEZS-112 (ZEN012) (tubulin inhibitor)

205797  ||  Macimorelin (AEZS-130 (EP-1572) (growth hormone agonist)

205799  ||   AF802 (CH5424802) (ALK inhibitor)

200500  ||  Afatinib (BIBW-2992 ) (EGFR inhibitor)

200120  ||  Afimoxifene (selective estrogen receptor modulator)

200123  ||  AFP-464 (aryl hydrocarbon receptor agonist)

205810  ||  AFX-2 (North American ginseng extract)

204240  ||  AFX-9901 (anti-angiogenic agent)

204250  ||  AG-013 (Trefoil Factor)

200125  ||  AG-24322 (CDK inhibitor)

200121  ||  AG-490 (EGFR and JAK inhibitor)

204260  ||  AI-850 (cremaphor-free formulation of paclitaxel)

205942  ||  AKN-028 (FLT3/KIT kinase inhibitor)

200127  ||  AKR-501 (thrombopoietin receptor agonist)

200130  ||  Alanosine (antimetabolic agent; adenylosuccinate synthetase inhibitor)

200131  ||  ALB-109564 ( tubulin inhibitor; antimitotic agent)

200133  ||  Alendronate sodium (geranyltranstransferase inhibitor)

201931  ||  Alisertib (MLN-8237) (Aurora A kinase inhibitor)

205943  ||  Almurtide (CGP-11637) (immunostimulating agent)

200170  ||  Alvespimycin (Hsp90 inhibitor)

200180  ||  Alvocidib (Flavopiridol) (CDK inhibitor)

200182  ||  Ametantrone (DNA intercalator)

200185  ||  AMG-208 (c-Met inhibitor)

204310  ||  AMG-319 (PI3 Kinase inhibitor  )

204320  ||  AMG-337 (c-Met inhibitor)

205898  ||  AMG-458 (c-Met inhibitor)

204370  ||  AMG-900 (inhibitor of Aurora kinases A, B, and C.)

205944  ||  Aminocamptothecin (topoisomerase I inhibitor)

200200  ||  Amonafide dihydrohloride (topoisomerase II inhibitor)

200210  ||  Amonafide malate (AS-1413) (topoisomerase II inhibitor)

200220  ||  Amrubicin (anthracycline; DNA intercalactor; topoisomerase II inhibitor)

205769  ||  Amsalog (topoisomerase II inhibitor)

200720  ||  Amsilarotene (TAC-101) (oral synthetic retinoid)

201950  ||  Amuvatinib (MP-470) (Multitargeted receptor tyrosine kinase inhibitor)

204371  ||  AN-207 (LHRH doxorubicin conjugate)

200252  ||  AN-2728 (PDE4 inhibitor)

200257  ||  ANA-773 (TLR7 agonist)

200230  ||  Anamorelin (RC1291) (ghrelin receptor agonist)

205811  ||  Aneustat (OMN54) (mixture of extracts from three commonly used Chinese medicine components; Ganoderma lucidum, Salvia miltiorrhiza and Scutellaria barbata)

200240  ||  Annamycin (DNA intercalactor; topoisomerase II inhibitor)

200250  ||  ANX-510 (thymidylate synthase inhibitor)

204380  ||  ANX-514 (docetaxel new formulation)

205899  ||  AP1903 (Dimerizer drug)

200255  ||  AP5346 (DACH polymer platinate )

205765  ||  AP-26113 (dual ALK and EGFR inhibitor)

200135  ||  Apatinib (VEGFR inhibitor)

200140  ||  Apaziquone (bioreductive prodrug, hypoxia toxic agent)

205812  ||  APC-100 (androgen antagonist)

205813  ||  APC-200 (ROS inhibitor)

205814  ||  APC-300 (signal transduction inhibitor)

200270  ||  Daporinad (APO-866) (FK866) (NAMPT inhibitor)

205945  ||  APR-246 (p53 activator)

205894  ||  Apremilast (PDE4 inhibitor)

200273  ||  Apricoxib (COX-2 inhibitor)

200272  ||  AR-12 (OSU-03012) (PDK-1 inhibitor)

200275  ||  AR-42 (HDAC inhibitor)

205815  ||  Armodafinil (CNS stimulantor)

204420  ||  ARN-509 (androgen receptor antagonist)

206041  ||  ARN-810 (selective estrogen receptor degrader, SERD)

200280  ||  Aroplatin (DNA crosslinking agent)

205946  ||  ARQ-087 (pan FGFR inhibitor)

200281  ||  ARQ-092 (AKT inhibitor)

205947  ||  ARQ-171 (E2F1 pathway activator)

200284  ||  ARQ-501 ( R1668,  beta-lapachone) (DNA damage checkpoint pathway activator)

204430  ||  ARQ-621 (Eg5 inhibitor)

204440  ||  ARQ-736 (BRAF Inhibitor)

205816  ||  ARQ-761 (beta-lapachone prodrug; DNA damage checkpoint pathway activator)

200290  ||  ARRY-300 (MEK inhibitor)

200291  ||  ARRY-380 (HER2 inhibitor)

205900  ||  ARRY-382 (cFMS inhibitor)

200292  ||  ARRY-520 (KSP inhibitor)

200294  ||  ARRY-614 (p38 and Tie2 kinase  inhibitor)

200310  ||  Arzoxifene (selective estrogen receptor modulators (SERMs))

205817  ||  AS101 (interleukin-10 inhibitor)

200296  ||  AS-605240 (PI3K Inhibitor)

200297  ||  AS703026 (MSC1936369B) (MEK 1/2 inhibitor)

205859  ||  AS703988 (MSC201510B) (MEK 1/2 inhibitor)

204450  ||  ASP-3026 (ALK inhibitor)

205818  ||  ASP-9521 (17βHSD5 inhibitor)

200314  ||  AT-101(Gossypol acetic acid) (Bcl-2 inhibitor)

205884  ||  AT13148 (AGC kinase inhibitor; PKB inhibitor)

200317  ||  AT-13387 (Hsp90 inhibitor)

204460  ||  AT-406 (IAP inhibitor)

200320  ||  AT-7519 (CDK inhibitor)

200322  ||  AT-9283 (multiple kinase inhibitor)

205786  ||  Ataluren (PTC124) (CFTR-G542X nonsense allele inhibitor)

200330  ||  Atamestane (aromatase inhibitor)

200340  ||  Atiprimod (STAT3 inhibitor)

200350  ||  ATN-161 (integrin alpha5beta1 inhibitor)

200360  ||  ATN-224 (SOD1 inhibitor)

200370  ||  Atrasentan (ABT-627) (endothelin A receptor antagonist)

200371  ||  AUY-922 (NVP-AUY922,  VER-52296) (Hsp90 inhibitor)

204480  ||  AVL-292 (BTK inhibitor)

200390  ||  AVN-944 (VX-944) (IMPDH inhibitor)

200400  ||  Axitinib (VEGFR inhibitor)

205948  ||  AZD-0424 (Src/Abl kinase inhibitor)

200421  ||  AZD1152-HQPA (Aurora B inhibitor)

205763  ||  AZD-1208 (pan-PIM kinase inhibitor)

204510  ||  AZD-1480 (JAK2 inhibitor)

204520  ||  AZD-2014 (mTOR inhibitor）

204530  ||  AZD-2461 (PARP inhibitor)

206039  ||  AZD-3463 (ALK/IGF1R inhibitor)

204540  ||  AZD-3514

206040  ||  AZD-3965 (MCT1 inhibitor)

204550  ||  AZD-4547 (pan-FGFR inhibitor)

200422  ||  AZD-4769 (EGFR tyrosine kinase inhibitor)

200424  ||  AZD-4877 (KSP inhibitor)

200425  ||  AZD-4992

205669  ||  AZD-5363 (PKB/Akt inhibitor)

200426  ||  AZD-5438 (CDK Inhibitor)

200427  ||  AZD-6126 (tubulin  Inhibitor)

200310  ||  AZD-6918

205820  ||  AZD-7451 ( TRK inhibitor)

200311  ||  AZD-7762 (checkpoint kinase inhibitor)

200312  ||  AZD-8055 (mTOR inhibitor)

200313  ||  AZD-8330 (ARRY-704)

200298  ||  AZD-8931 (HER1and HER2 inhibitor)

206042  ||  AZD9291

200315  ||  AZM-475271 (Src tyrosine kinase inhibitor)

200316  ||  Bafetinib (INNO-406) (Bcr/Abl inhibitor)

205821  ||  BAL101553 (microtubulin inhibitor)

205822  ||  BAL27862  (microtubulin inhibitor)

200430  ||  Banoxantrone (hypoxia toxic agent)

200420  ||  Barasertib (AZD-1152) (Aurora B inhibitor)

202530  ||  Bardoxolone methyl (RTA402) (antioxidant inflammation modulator)

205893  ||  Baricitinib (INCB28050, LY3009104) (JAK1 and JAK2 inhibitor)

200440  ||  Batabulin sodium (tubulin  inhibitor)

200442  ||  Batimastat (MMP Inhibitor)

204560  ||  BAY 10-00394 ( (CDK inhibitor)

205923  ||  BAY 10-82439 (PI3Kα/β inhibitor)

205949  ||  BAY 56-3722 (water soluble camptothecin derivative)

204570  ||  BAY 80-6946 (PI3K inhibitor)

205901  ||  BAY 87-2243 (HIF-1ἀ pathway inhibitor)

204590  ||  BAY 94-9392 (F18 tumor PET imaging agent)

205902  ||  BBI503 (cancer stemness kinase inhibitor)

204620  ||  BBI-608 (Cancer cell stemness inhibitor)

200450  ||  Becatecarin (DNA intercalator)

200455  ||  Beclometasone dipropionate (potent glucocorticoid steroid)

200460  ||  Belinostat (HDAC inhibitor)

205929  ||  Beloranib (CDK-732, ZGN-433) (MetAP-2 inhibitor)

200461  ||  Belotecan (camptothecin derivative; topoisomerase I inhibitor)

200470  ||  Bendamustine HCl (DNA alkylator)

200480  ||  Beraprost (prostacyclin derivative)

200490  ||  Berubicin (topoisomerase II inhibitor; anthracycline derivative)

200160  ||  Betulinic acid (  ALS357) (melanoma-specific cytotoxic agent)

204920  ||  Bevonium methylsulfate (also see CG-201) ( hCG inhibitor)

200491  ||  BEZ235 ( NVP-BEZ235) (PI3K inhibitor)

204790  ||  Bezielle (BZL-101) (extract of plant Scutellaria barbata; apoptosis inducer)

205888  ||  BGC-638 (thymidylate synthase inhibitor)

209490  ||  BGC-945 (ONX-0801) (thymidylate synthase inhibitor)

204640  ||  BGJ-398 (pan FGFR kinase inhibitor)

200492  ||  BGT226 (NPV-BGT226) (PI3K inhibitor)

200493  ||  BI-2536 (Polo-like kinase 1 inhibitor)

204670  ||  BI-811283 (Aurora kinase inhibitor)

200495  ||  BI-831266 (temporally not available)

205823  ||  BI-836825 (temporally not available)

205824  ||  BI-847325 (temporally not available)

205825  ||  BI-853520 (PTK2 inhibitor, focal adhesion kinase inhibitor)

200505  ||  BIIB-021 (CNF2024) (HSP90 inhibitor)

204676  ||  BIIB028  (Hsp90 inhibitor)

205826  ||  BIND-014 (PSMA-targeted docetaxel nanoparticles)

200515  ||  BIX-02188 (MEK5 inhibitor)

205951  ||  Bizelesin (DNA-interactive agent)

204690  ||  BKM-120 (PI3K inhibitor)

205878  ||  BKT140 (CXCR4 antagonist )

204710  ||  BMN-673 (PARP inhibitor)

205952  ||  BMS-214662 (Farnesyltransferase inhibitor)

200520  ||  BMS-275183 (paciltaxel analogue, tubulin inhibitor)

200524  ||  BMS-536924 (IGF-IR kinase inhibitor)

200531  ||  BMS-641988  (androgen receptor (AR) antagonist)

200533  ||  BMS-690514 (VEGFR inhibitor; HER inhibitor)

200534  ||  BMS-754807 (IGF-1R inhibitor)

200527  ||  BMS-777607 (Met tyrosine kinase inhibitor)

200535  ||  BMS-833923 (XL-139)

205768  ||  BMS-863233 (XL-413) (CDC7 kinase inhibitor)

205767  ||  BMS-911543 (JAK2 inhibitor)

205827  ||  BMS-906024 (NOTCH inhibitor)

204740  ||  BMS-936558 (an anti-programmed death-1 (MDX-1106))

204750  ||  BMS-936559 (an anti-programmed death-1)

204760  ||  BNC-105 (Vascular disrupting agent, tubulin polymerization inhibitor)

205749  ||  BNC105P (Vascular disrupting agent, tubulin polymerization inhibitor)

200560  ||  Bosutinib (Abl and Src  inhibitor)

200561  ||  BQS-481

205953  ||  Brequidar (dihydroorotate dehydrogenase inhibitor)

200569  ||  Brivanib (VEGFR2 inhibitor)

200570  ||  Brivanib alaninate (VEGFR2 inhibitor)

202520  ||  Brivudin (RP-101)

200580  ||  Brostallicin

200584  ||  BTZ043

204780  ||  BYL719 (PI3K inhbitor)

200585  ||  Cabazitaxel (XRP-6258) (tubulin inhibitor)

200595  ||  Cabozantinib ( XL-184) (VEGFR2, Met, FLT3, Tie2, Kit and Ret inhibitor)

200586  ||  CAL-101 (PI3K inhibitor)

200600  ||  Canertinib

200610  ||  Canfosfamide

201453  ||  Capesaris (GTX-758) (estrogen receptor (ER) alpha agonist)

200620  ||  Carbendazim

204830  ||  Carboxyamidotriazole orotate  (CTO)

200630  ||  Carfilzomib (proteasome inhibitor)

200650  ||  Casopitant mesylate

204840  ||  CB-1400 (Not Available)

204860  ||  CBP-501

205954  ||  CBT-1 (MDR modulator)

205829  ||  CC-115 (DNA-PK/TOR kinase inhibitor)

205830  ||  CC-122 (Pleiotropic Pathway Modulator)

205831  ||  CC-1088 (selective cytokine inhibitory drug; phosphodiesterase-4 inhibitor)

205955  ||  CC-11006 (immunomodulatory agent)

204870  ||  CC-223（mTOR inhibitor）

200651  ||  CC-401

200670  ||  CC-8490

205877  ||  CCX2206 (CXCR7-specific inhibitor)

200690  ||  Cediranib (AZD2171) (VEGF inhibitor)

200694  ||  Celastrol (HSP90 inhibitor)

200700  ||  Celecoxib

200710  ||  Cemadotin

200716  ||  CEP-7055

204910  ||  CEP-9722 (PARP inhibitor)

200712  ||  CEP-11981 (VEGFR inhibitor)

200713  ||  CEP-18770 (proteasome inhibitor)

205903  ||  CEP-32496 (BRAF kinase inhibitor)

205876  ||  Cepharanthine (TNF-α inhibitor)

200721  ||  Cerovive (NXY-059)

200730  ||  Cevipabulin (antimicrotubule agent)

200740  ||  CF-101

205956  ||  CFG920 (CYP17 inhibitor)

200750  ||  CGC-11047 (PG-11047)

205957  ||  CGM097 (p53/HDM2 interaction inhibitor)

200752  ||  CGS-21680 (adenosine A2A receptor agonist)

205747  ||  CH5132799  (PI3K inhibitor)

200755  ||  Chelerythrine chloride

204930  ||  Chidamide  (CS055;  HBI-8000)

200770  ||  CHIR-265 (also  see: RAF-265)

200774  ||  CHIR-99021

205770  ||  CHR-2845 (HDAC inhibitor)

205771  ||  CHR-3996 (HDAC inhibitor)

200776  ||  CHS-828 (NAD inhibitor)

205921  ||  CI-994 (HDAC inhibitor)

200771  ||  CI-1040 (also  see: PD184352)

200780  ||  Cilengitide (αVβ3/αVβ5 integrin inhibitor )

205832  ||  Cipatinib (oral tyrosine kinase inhibitor)

200781  ||  CJ-15161

205612  ||  CKI27 (RG7304) (MEK inhibitor)

205833  ||  CKD-516 (microtubulin inhibitor)

200790  ||  Clodronate disodium

204940  ||  CLR-1404

200791  ||  CNDO-101

204970  ||  CO-101 (Gemcitabine elaidate; CP-4126) (antimetabolite agent)

205796  ||  CO-1686 (AVL-301) (EGFR inhibitor)

200793  ||  Cordycepin (also  see: OVI-123)

200810  ||  CP-547632 (VEGFR-2 inhibitor)

200820  ||  CP-724714 (HER2 inhibitor)

200823  ||  CPI-613 (metabolic inhibitor)

204990  ||  CPX-1  (formulation of Irinotecan + Floxuridine)

205010  ||  CPX-351 (formulation of cytarabine + daunorubicin)

205020  ||  Crenolanib (CP-868596) (PDGFR inhibitor)

202222  ||  Crizotinib (PF-2341066) (tyrosine kinase inhibitor)

205030  ||  CRLX-101

200831  ||  Crolibulin (EPC2407) (tubulin inhibitor)

200841  ||  CUDC-101 (HDAC, EGFR and HER2 inhibitor)

205924  ||  CUDC-907  (a dual PI3K and HDAC inhibitor)

200842  ||  CVT-6883 (A2B adenosine antagonist)

205834  ||  CWP232204 (Wnt signaling inhibitor)

205904  ||  CWP232291 (Sam68 modulator)

200848  ||  CX-5461 (RNA polymerase I Inhibitor)

200844  ||  CYC-116 (Aurora kinase/VEGFR2 inhibitor)

200786  ||  CYT-387 (JAK inhibitor)

205959  ||  Cytochlor (radio-sensitizing agent)

205748  ||  Lexibulin (CYT997) (Vascular disrupting agent)

205653  ||  D-3263

205479  ||  Dabrafenib (GSK-2118436) (B-RAF inhibitor)

200845  ||  Dacinostat (NVP-LAQ824)

205576  ||  Dacomitinib (PF-00299804) (EGFR inhibitor)

205960  ||  Daniquidone (Batracylin) (DNA topoisomerase inhibitor)

200846  ||  Danusertib (PHA-739358) (Aurora kinase inhibitor)

200850  ||  Darinaparsin (ZIO-101)

200851  ||  DCC-2036 (BCR-ABL inhibitor)

205737  ||  Debio-0932 (CUDC-305) (Hsp90 inhibitor)

100255  ||  Degarelix acetate

200890  ||  Denibulin (MN-029) (microtubule inhibitor; vascular-disrupting agent)

201000  ||  Dexmethylphenidate (NDRI inhibitor)

206008  ||  Diazepinomicin (TLN-4601) (RAS/RAF/MAPK inhibitor)

200900  ||  Diethylnorspermine

201020  ||  Diflomotecan

205999  ||  Dilmapimod (SB-681323) (GW-681323)(p38 MAPK inhibitor)

201030  ||  Dimesna

202572  ||  Dinaciclib (SCH-727965, PS-095760) (CDK inhibitor)

200880  ||  DMPEN(4-demethylpenclomedine) (alkylation agent)

201060  ||  Docosahexaenoic acid

201065  ||  Dofequidar (P-glycoprotein inhibitor; MDR inhibitor; sphingomyelin synthase inhibitor)

201040  ||  Doramapimod (p38 MAPK inhibitor)

200760  ||  Dovitinib (TKI-258,  CHIR258) (fibroblast growth factor receptor 3 (FGFR3) inhibitor)

205835  ||  DS-2248 (Hsp90 inhibitor)

205961  ||  DS-3078a (TORC1/2 kinase inhibitor)

205836  ||  DS-7423 (PI3K/mTOR kinase inhibitor)

201070  ||  Dutasteride

205837  ||  E-3810 (VEGFR/FGFR dual kinase inhibitor)

201071  ||  E6201 ( MEK-1/MEKK-1 inhibitor)

205150  ||  E7016 (PARP inhibitor)

201072  ||  Golvatinib (E7050) ( c-Met/VEGFR kinase inhibitor)

205882  ||  E7449: (PARP inhibitor)

201090  ||  E7820 (angiogenesis inhibitor)

201100  ||  E7974

205170  ||  EC-0225

205180  ||  EC-0489

205190  ||  EC-145

205210  ||  EC-17

201150  ||  Edatrexate

201160  ||  Edotecarin (PHA-782615; J-107088; ED-749) (topoisomerase inhibitor)

201180  ||  Efaproxiral (radiosensitizer)

205260  ||  Eflornithine (CPP-1X)

201190  ||  Elacridar (P-glycoprotein inhibitor)

201195  ||  Elacytarabine (antimetabolite agent)

201200  ||  Elagolix ( NBI-56418)

201210  ||  Elesclomol (HSP-90 Inhibitor)

201220  ||  Elinafide (DNA intercalator)

202300  ||  Elisidepsin (PM-02734)

205828  ||  Elomotecan (BN-80927) (topoisomerase inhibitor)

201230  ||  Elsamitrucin (DNA intercalator)

201240  ||  Eltrombopag (thrombopoietin receptor agonist)

205330  ||  EMD-1204831 (c-MET inhibitor)

201245  ||  EMD-1214063 (c-Met inhibitor)

206035  ||  EMD534085 (Kinesin inhibitor)

201250  ||  Eniluracil (dihydropyrimidine dehydrogenase inhibitor)

201260  ||  ENMD-1198 (antimitotic agent)

201264  ||  ENMD-2076 (Aurora kinase inhibitor)

201266  ||  Entinostat (MS-275,  SNDX-275) (HDAC inhibitor)

201821  ||  Enzalutamide (MDV3100) (selective androgen receptor modulator)

201270  ||  Enzastaurin (LY317615) (protein kinase C beta inhibitor)

201275  ||  Epofolate (BMS-753493) (folate receptor-targeting antimitotic agent)

201280  ||  Epothilone D ) (tubulin inhibitor)

205892  ||  EPZ-5676 (DOT1L inhibitor and HMT inhibitor)

201290  ||  Eribulin mesylate (E7389) (tubulin inhibitor)

205510  ||  Erismodegib (LDE225, NVP-LDE225) (Smo antagonist)

201300  ||  ES285

201310  ||  Etalocib (LY293111) (LTB4 receptor antagonist)

206031  ||  Etanidazole (SR-2508) (bioreductive drug)

205230  ||  Etarfolatide (EC-20) (tumor imaging agent)

201320  ||  Ethonafide

201330  ||  Ethynylcytidine

100335  ||  Everolimus

201340  ||  Exatecan (topoisomerase inhibitor)

201350  ||  Exherin

201354  ||  Exisulind

201360  ||  Ezatiostat (glutathione S-transferase P1-1 (GSTP1-1) inhibitor)

205962  ||  Fadrozole (aromatase inhibitor)

205950  ||  Falnidamol ((EGFR inhibitor)

205935  ||  Famitinib (multi-targeted RTK inhibitor)

205963  ||  Fazarabine (Kymarabine) (DNA synthesis inhibitor)

205430  ||  Fenretinide (RAR agonist)

205450  ||  Finasteride

205380  ||  Firtecan pegol (EZN-2208) (Pegylated SN-38, drug conjugate)

205460  ||  Fluciclatide F-18

201380  ||  Fludarabine

205905  ||  Fluorapacin

201372  ||  Foretinib (XL880, SK1363089, GSK089, EXEL-2880) (MET/VEGFR2 inhibitor)

201390  ||  Forodesine

205461  ||  Fosaprepitant  (antiemetic agent)

200800  ||  Fosbretabulin (combretastatinA-4phosphate, CA4P) (vascular disrupting agent)

205965  ||  Fosquidone (topoisomerase inhibitor)

201393  ||  Fostamatinib (R788) (Syk kinase inhibitor)

205465  ||  FT-1050 (Stem Cell Modulator)

205646  ||  Galeterone (TOK-001)

202703  ||  Ganetespib (STA-9090) (Hsp90 inhibitor)

205746  ||  GDC-0032 (PI3K inhibitor)

205467  ||  GDC-0068 (AKT  inhibitor)

205764  ||  GDC-0152 (IAP inhibitor, Smac mimetic)

205839  ||  GDC-0349

205840  ||  GDC-0425 (RG7602) (ChK-1 inhibitor)

205841  ||  GDC-0575 (ChK1 selective inhibitor)

205772  ||  GDC-0623 (MEK inhibitor)

205468  ||  GDC-0917 (IAP inhibitor)

201395  ||  GDC-0941 (PI3K inhibitor)

203185  ||  GDC-0973 (XL518) (MEK inhibitor)

205470  ||  GDC-0980 (RG7422) ( PI3 kinase/mTOR inhibitor)

205471  ||  GENZ-644282 (A non-camptothecin inhibitor of topoisomerase I)

205922  ||  Geldanamycin (HSP 90 inhibitor)

205798  ||  GFB-204 (VEGFR and PDGFR inhibitor)

205472  ||  GGTI-2418 (geranylgeranyltransferase I inhibitor)

201410  ||  Gimatecan (topoisomerase inhibtor)

205774  ||  Givinostat (ITF2357) (HDAC inhibitor)

205842  ||  GLPG0187 (integrin receptor antagonist)

201420  ||  Glufosfamide

205843  ||  GO-203-2C (MUC1-targeted peptide)

201422  ||  Golotimod

201430  ||  Gossypol (Bcl-2 inhibitor)

201436  ||  GPI-15427

201440  ||  GPX100 (anthracycline, DNA intercalator)

201450  ||  GPX150 (anthracycline, DNA intercalator)

205475  ||  GRN-1005 (ANG-1005) (paclitaxel conjugate, microtube inhibitor)

201452  ||  GS-9219

205966  ||  GS-9820 (p110beta/delta PI3K Inhibitor)

205739  ||  GSK-1059615 （mTOR inhibitor）

205477  ||  GSK-1070916A (Aurora B/C kinase inhibitor)

205478  ||  GSK-2110183 (AKT inhibitor)

205480  ||  GSK-2126458 (PI3K inhibitor, mTOR inhibitor)

205481  ||  GSK-2141795 (Akt inhibitor)

205482  ||  GSK-2256098

205483  ||  GSK-2401502

205484  ||  GSK-2586881 (APN01)

205844  ||  GSK-2636771 (PI3K inhibitor)

205667  ||  GSK-461364  (PLK inhibitor)

205697  ||  GSK-525762 (BET inhibitor)

205670  ||  GSK-690693 (pan-Akt kinase inhibitor)

205036  ||  GSK-923295 (Kinesin inhibitor)

205766  ||  Gusperimus (immunosuppressant agent)

201460  ||  HA14-1

205968  ||  Halofuginone

205485  ||  HE-3235

205845  ||  Henatinib (multitargeted tyrosine kinase inhibitor)

201466  ||  Hesperadin

401510  ||  HM30181 (MDR1 inhibitor)

205969  ||  HM61713 (EGFR inhibitor)

205846  ||  HM781-36B (irreversible pan-HER inhibitor)

201480  ||  HMN-176 (PLK-1 inhibitor)

201490  ||  HMN-214 (PLK-1 inhibitor)

205486  ||  HQK-1004

205487  ||  HSP-990 (HSP inhibitor)

205735  ||  Hycanthone (Topoisomerase inhibitor, DNA intercalator)

201495  ||  Hypothemycin

205879  ||  Laniquidar (R101933) (Oral P-glycoprotein Inhibitor)

202171  ||  Ibrutinib (PCI-32765) (BTK inhibitor)

201684  ||  Ibutamoren

205847  ||  Icotinib (EGFR inhibitor)

205880  ||  Idoxifene (estrogen antagonist)

205489  ||  Imetelstat  (GRN-163L)

201500  ||  Imexon (caspase inhibitor)

205886  ||  IMMU-132 (antibody-SN38 conjugate)

201510  ||  Imidazoacridone

205492  ||  IMO-2055 (EMD1201081)

205494  ||  INC280 (INCB-028060) (c-MET inhibitor, RTK inhibitor)

205493  ||  INCB024360 (IDO1 inhibitor)

201520  ||  Incyclinide

201530  ||  Indibulin (ZIO-301) (tubulin inhibitor)

206023  ||  Indirubin (CDK inhibitor)

201540  ||  Indisulam (carbonic anhydrase inhbitor)

205971  ||  Indomethacin (COX inhibitor)

201545  ||  Ingenol Mebutate (PEP005)

200582  ||  Iniparib (BSI-201) (PARP inhibitor)

201550  ||  INNO-206 (DNA intercalating agent)

201561  ||  INO-1001

205250  ||  Inolitazone (CS-7017, Efatutazone )

201562  ||  INSM-18

200496  ||  Nintedanib  ( BIBF-1120)  (VEGFR inhibitor)

201570  ||  Iobenguane

205496  ||  Ioflubenzamide I-131 (MIP-1145)

205744  ||  IPI-145 (INK-1197) (PI3K inhibitor)

205773  ||  IPI-269609 (Hedgehog pathway inhibitor)

201571  ||  IPI-493

201580  ||  Irofulven

200550  ||  Irosustat (STX64, BN83495)

205906  ||  IRX4204 (RXR agonist)

205907  ||  IRX4310 (pan-RAR antagonist)

201590  ||  Isatoribine (toll-like receptor 7 (TLR-7) agonist)

205848  ||  Iso-Fludelone (microtubulin inhibitor)

201600  ||  Ispinesib

201610  ||  Ixabepilone

205541  ||  Ixazomib (MLN-9708) (the first oral proteasome inhibitor)

201611  ||  JI-101

201613  ||  JNJ-26483327

201615  ||  JNJ-38877605 (tyrosine kinase inhibitor)

205972  ||  JNJ-40346527 (FMS inhibitor)

205973  ||  JNJ-42756493 (FGFR inhibitor)

205849  ||  JNS002 (Pegylated liposomal doxorubicin)

201620  ||  Kahalalide F

201630  ||  Karenitecin (Cositecan,  BNP-1350).

201640  ||  Ketamine

205891  ||  Kevetrin (Protein p53 activator)

201650  ||  KOS-1584 (R1645)

206021  ||  KP1019 (ruthenium metastasis inhibitor)

205883  ||  KPT-330 (Selective Inhibitor of Nuclear Export, SINE)

201660  ||  KRN5500

205868  ||  KRN7000 (RGI-2001) (immunomodulator)

205775  ||  KRP-203 (Sphingosine-1-phosphate receptor agonist)

201670  ||  KRX-0402

203060  ||  KRX-0601(also  see UCN-01)

205776  ||  KU-0063794 (mTOR inhibitor)

206034  ||  KU-2285 (hypoxic cell sensitizer)

201681  ||  KU-55933

201684  ||  KW-2449

205908  ||  KW-2450 (IGF-1R/IR inhibitor)

205506  ||  KW-2478 (Hsp90 inhibitor)

205927  ||  KX-01 ( Src kinase inhibitor)

201686  ||  KX2-391 (rc kinase inhibitor)

205974 ||   L-377202 (doxorubicin conjugate)

205508  ||  Lansoprazole

201705  ||  Laromustine(VNP40101M)

201710  ||  Larotaxel (XRP9881)

201720  ||  Lasofoxifene

205909  ||  LCI699 (aldosterone synthase inhibitor)

205509  ||  LCL-161

205511  ||  LDK-378 (ALK inhibitor)

205512  ||  LE-DT (Liposome Encapsulated Docetaxel)

205993  ||  Ledoxantrone (topoisomerase II inhibitor)

205513  ||  LEE-011

201724  ||  Lemuteporfin (QLT-0074) (PDT photosensitizer)

201080  ||  lenvatinib (E7080)

205514  ||  LEP-ETU (liposomal paclitaxel, PNU-93914)

205515  ||  LEQ-506

205975  ||  Lerisetron (3,5-HT3) receptor antagonist)

201730  ||  Lestaurtinib

205895  ||  Letaxaban (TAK-442) (Factor Xa inhibitor)

100542  ||  Levoleucovorin Calcium

201741  ||  LGD-4665

205850  ||  LGH447 (PIM inhibitor)

205851  ||  LGK-974 (Porcupine inhibitor)

205852  ||  LGX818 (Raf kinase inhibitor)

205976  ||  Liarozole (retinoic acid metabolism blocking agent)

200060  ||  Linifanib ( ABT869) (RTK inhibitor)

202096  ||  Linsitnib (OSI-906) (IGF-1R inhibitor)

205521  ||  Litronesib (aslo see: LY2523355)

201750  ||  Lomeguatrib

205977  ||  Lometrexol (GARFT inhibitor; anti-metabolizing agent)

201760  ||  Lonafarnib (farnesyl transferase inhibitor)

205910  ||  Lonaprisan (progesterone receptor antagonist)

205517  ||  LOR-253 (MTF-1 inhibitor)

205853  ||  LOR-500 (MELK inhibitor)

206028  ||  Losoxantrone (DNA intercalator, bioreductive drug)

201761  ||  LP-261

201780  ||  Lucanthone (Topoisomerase inhibitor, DNA intercalator)

205594  ||  Lurbinectedin (PM-01183) (DNA minor groove-binding agent)

205783  ||  Lurtotecan (OSI-221; NX221) (topoisomerase I inhibitor)

205518  ||  LY2090314 (GSK-3 inhibitor)

205520  ||  LY2157299 (TGF-βR inhibitor)

205854  ||  LY2228820 (p38MAPK inhibitor)

201792  ||  LY2334737 (antimetabolite agent)

205925  ||  LY2457546 (multikinase inhibitor)

205522  ||  LY2584702

201794  ||  Rabusertib (LY2603618) (CHK2 inhibitor)

205523  ||  LY2606368

205524  ||  LY2624587 (not available)

205525  ||  LY2780301 (AKT inhibitor)

206032  ||  LY2784544 (JAK inhibitor)

205526  ||  LY2801653 (c-MET inhibitor) 

205911  ||  LY2835219 (CDK inhibitor)

205527  ||  LY2874455 (FGFR inhibitor)

205528  ||  LY2875358 (anti-c-MET monoclonal antibody)

201795  ||  LY294002 (PI3K inhibitor)

205529  ||  LY2940680

205855  ||  LY3007113 (p38 MAPK inhibitor)

201800  ||  M40403

205912  ||  Macitentan (endothelin receptor antagonist)

205978  ||  Mafosfamide (DNA cross-linking agent)

201802  ||  Marimastat (BB-2516)

202031  ||  Marizomib (NPI-0052) (proteasome inhibitor)

201804  ||  Masitinib (AB1010) (tyrosine kinase inhibitor)

205741  ||  Maytansine (microtubule inhibitor)

201810  ||  Imisopansem manganese (MB07133)

205782  ||  ME-143 (NV-143) (NADH oxidase inhibitor)

205856  ||  ME-344 (mTOR1/2 kinase inhibitor)

205531  ||  MEK-162 (ARRY-162) (MEK1/2  inhibitor)

205650  ||  Methoxyamine (TRC102) (DNA base excision repair (BER) inhibitor)

205533  ||  Methyl aminolevulinate  (PDT photosensitizer)

205671  ||  MG-516 (multi-targeted kinase inhibitor)

201841  ||  MGCD-265 (multitargeted tyrosine kinase inhibitor)

201850  ||  Midostaurin (PKC412)

201860  ||  Mifamurtide (L-MTP-PE. MTP-PE) (immunomodulatory agent)

201870  ||  Mifepristone

201880  ||  Milataxel

202233  ||  Milciclib (PHA-848125) (CDK inhibitor and TRKA inhibitor)

201890  ||  Miltefosine

205536  ||  MIP-1095

205979  ||  Mitoguazone (SAMD inhibitor)

205980  ||  Mivobulin isethionate (microtubule inhibitor)

201891  ||  MK-0429 (ανβ3 Integrin Inhibitor)

201910  ||  MK-0731 (KSP inhibitor)

201911  ||  MK-0752 (notch inhibitor)

205537  ||  MK-1496 (Polo-like kinase 1 inhibitor)

201912  ||  MK-1775 (WEE inhibitor)

201913  ||  MK-2206 (Akt inhibitor)

201914  ||  MK-2461 (Multitargeted Kinase Inhibitor)

201915  ||  MK-4101 (not available)

201916  ||  MK-4827 (PARP inhibitor)

201917  ||  MK-5108 (VX-689) ( Aurora-A kinase inhibitor)

201918  ||  MK-8033 (c-MET inhibitor)

201920  ||  MKC-1

201922  ||  MKI-833

205495  ||  MLN0128 (INK-128) (mTOR inhibitor)

205743  ||  MLN1117 (INK-1117) (PI3K inhibitor)

205857  ||  MLN-2238 (oral proteasome inhibitor, metabolite of MLN9708)

205777  ||  MLN-2480 (Raf kinase inhibitor)

201924  ||  MLN-4924 (NAE inhibitor)

201930  ||  MLN-8054 (aurora kinase inhibitor)

205858  ||  MM-151 (EGFR  inhibitor)

205720  ||  MM-302 (HER2-targeted liposomal doxorubicin)

205543  ||  MM-398 (irinotecan nanotherapy)

201932  ||  MN-201

201933  ||  Mocetinostat (MGCD-0103) (HDAC inhibitor)

201934  ||  Motesanib (AMG-706) (tyrosine kinase inhibitor)

201940  ||  Motexafin gadolinium (PDT photosensitizer, radiosensitizer)

201942  ||  Motexafin lutetium (PDT photosensitizer, radiosensitizer)

201944  ||  MP-412 (AV-412) (EGFR/HER2 tyrosine kinase inhibitor)

201951  ||  MPC-2130

205544  ||  MPC-3100 (Hsp90 inhibitor)

205885  ||  MRK 003 (γ-secretase inhibitor; Notch inhibitor, Hedgehog inhibitor)

205545  ||  MRX-1024

201961  ||  MSX-122 (CXCR4 inhibitor)

205549  ||  Nabiximols

206020  ||  NAMI-A (ruthenium metastasis inhibitor)

201980  ||  NBI-42902

206017  ||  Nebentan (YM598) endothelin A receptor antagonist)

201824  ||  Nemorubicin

201470  ||  Neratinib (HKI272) (HER2 and EGFR inhibitor)

205981  ||  Netupitant (NK1 receptor antagonist)

205940  ||  Niclosamide (Stat inhibitor)

205934  ||  Nifurtimox

201990  ||  Nilotinib (Bcr-Abl inhibitor)

205860  ||  Nitroarginine (NG-nitro-L-arginine) (nitric oxide synthase inhibitor)

205551  ||  NK-012 (SN-38-PEG conjugate, camptotecin conjugate)

205740  ||  NKP-1339 (ruthenium-based transferrin targeting agent)

205742  ||  NKP-2235 (gallium-based small molecule)

205552  ||  NKTR-102

205553  ||  NKTR-105

202000  ||  NM-3 (isocoumarin)

205778  ||  NMS-1116354 (CDC7 kinase inhibitor)

205779  ||  NMS-1286937 (PLK1 inhibitor)

202010  ||  Nolatrexed

205556  ||  Norepinephrine

202020  ||  Noscapine (also see CB-3304)

202030  ||  NOV-002 (chemoprotective agent)

201970  ||  Novitoclax (ABT-263) (Bcl-2 Inhibitor)

205982  ||  NRX-19583 (RAR alpha agonist)

202041  ||  NRX-4204 (NRX19402) (retinoid X receptor (RXR) agonist)

205861  ||  NS-018 (JAK2/Src inhibitor)

205557  ||  NUC-1031 (a phosphoramidate ProTide)

205780  ||  NV-128 (mTOT inhibitor)

202050  ||  Obatoclax (   GX15-070) (BCL-2 Inhibitor)

202062  ||  Odanacatib (MK-0822) (protease inhibitor)

206043  ||  ODM-201 (androgen receptor inhibitor)

202064  ||  Oglufanide

200423  ||  Olaparib (AZD-2281) (PARP inhibitor)

202070  ||  Oleandrin (PBI-05204)

205913  ||  Oltipraz (chemopreventive agent)

202075  ||  Omacetaxine mepesuccinate (Homoharringtonine)

200380  ||  Ombrabulin (AVE8062) (tubulin inhibitor)

200385  ||  Omtriptolide

205563  ||  ON-013105

205914  ||  ONO-4059 (BTK inhibitor)

205983  ||  ONO-7746 (TPO receptor agonist )

202087  ||  ONT-093 (OC144-093) (P-glycoprotein pump inhibitor)

205625  ||  ONX 0805 (SB1578)

205565  ||  ONX-0912 (proteasome inhibitor)

205730  ||  ONX-0914 (immunoproteasome inhibitor)

205566  ||  OPB-31121 (STAT3 inhibitor)

205567  ||  OPB-51602 (STAT3 inhibitor)

205890  ||  OKN-007 (neuroprotective nitrone)

205984  ||  Ormaplatin (DNA alkylating agent)

202090  ||  Ortataxel (taxane microtube inhibitor)

200724  ||  Orteronel (TAK-700) (steroid 17alpha-monooxygenase inhibitor)

202094  ||  OSI-027 (mTOR inhibitor)

205569  ||  OSI-7904L (GS7904L, OVI-237 ) (inhibitor of thymidylate synthase)

202100  ||  OSI-930

202103  ||  Ostarine (MK-2866, GTX-024)

205985  ||  OTX008 (galectin-1 inhibitor)

205570  ||  OXi-4503

202110  ||  Ozarelix (also  see: SPI-153)

205936  ||  P7170 (PI3K, mTOR and ALK1 inhibitor)

202114  ||  P2045

202118  ||  P276-00 (DCK inhibitor)

205571  ||  PA799 (PI3K class I inhibitor)

206029  ||  PA-824 (bioreductive drug)

205932  ||  PAC-1 (procaspase activator)

202571  ||  Pacritinib (SB1518)

205760  ||  Padeliporfin (WST11, Stakel) (PDT photosensitizer)

202185  ||  Padoporfin   (Tookad) (PDT photosensitizer)

202130  ||  Palifosfamide (ZIO-201)

202133  ||  Palomid 529 (PI3K inhibitor; Akt inhibitor; mTOR inhibitor)

202151  ||  Panobinostat (NVP-LBH589; LBH589) (HDAC inhibitor)

205572  ||  Pasireotide (SOM-230) ( somatostatin receptor agonist)

202160  ||  Patupilone (EPO906)

202161  ||  Pazopanib (GW786034) (tyrosine kinase inhibitor )

205574  ||  PCI-27483 (factor VIIa inhibitor)

202172  ||  PD-0325901 (MEK inhibitor)

202173  ||  PD-0332991 (CDK Inhibitor)

202174  ||  PD-153035 (EGFR inhibitor)  

205915  ||  Pegdinetanib (VEGFR-2 inhibitor peptide)

202190  ||  Pelitinib (EKB569) (pan-ErbB tyrosine kinase inhibitor)

202200  ||  Pelitrexol (GARFT inhibitor) (glycinamide ribonucleotide formyltransferase)

205986  ||  Peretinoin (RAR agonist)

202220  ||  Perifosine (AKT Inhibitor)

205916  ||  PF-00337210 (VEGFR2 tyrosine kinase inhibitor)

202224  ||  PF-03084014

202223  ||  PF-03732010 (antibody drug, p-cadherin antagonist)

205581  ||  PF-03758309 (PAK4 inhibitor)

205987  ||  PF-03814735 (Aurora kinase inhibitor)

205988  ||  PF-04136309 (CCR2 antagonist)

202221  ||  PF-04217903 ( MET tyrosine kinase inhibitor)

205582  ||  PF-04449913

205583  ||  PF-04554878 (FAK inhibitor)

202226  ||  PF-04691502 (PI3K/mTOR inhibitor)

202227  ||  PF-0477736 (CHK inhibitor)

202228  ||  PF-0562271 (PF-562271; PF-00562271) (a FAK inhibitor)

202231  ||  PHA-665752 (c-MET inhibitor)

206024  ||  PHA-793887 (CDK inhibitor)

202180  ||  Phenoxodiol

202242  ||  Photochlor (PDT photosensitizer)

206022  ||  PH-797804 ( p38 MAP kinase inhibitor)

202234  ||  PHY-906

202235  ||  PI-103 (PI3K inhibitor, and mTOR inhibitor)

202230  ||  Picoplatin

205819  ||  Picropodophyllin (AXL1717) (IGF-1 receptor inhibitor)

202238  ||  PIK-75 (PI3K inhibitor)

206030  ||  Pimonidazole (bioreductive drug)

202240  ||  Pipendoxifene

205784  ||  Piroxantrone (topoisomerase II inhibitor)

205928  ||  Pivanex (AN-9) (HDAC inhibitor)

202250  ||  Pixantrone

205989  ||  PKI-179 (PI3Ka/mTOR inhibitor)

202255  ||  PKI-587 (PF-05212384) (Dual PI3 Kinase/mTOR Inhibitor)

202260  ||  Plerixafor

202270  ||  Plevitrexed (BGC-9331)

202040  ||  Plinabulin (NPI-2358)

200150  ||  Plitidepsin (Aplidine)

205592  ||  PLX-3397 (multitargeted tyrosine kinase inhibitor)

202272  ||  PLX-4720 (B-Raf inhibitor)

202290  ||  PM-00104

205595  ||  PM-060184

202301  ||  PN-401

205596  ||  PNT-2258 (an oligonucleotide therapeutic encapsulated within a SMARTICLES formulation).

205514  ||  PNU-93914 (liposomal paclitaxel, LEP-ETU)

205864  ||  POL6326 (CXCR4 inhibitor)

202302  ||  Polyphenon E

202310  ||  Pomalidomide

202320  ||  Ponatinib (AP-24534) (tyrosine kinase inhibitor)

202324  ||  PP242 (mTOR inhibitor)

202330  ||  PPI-2458

202331  ||  PR-104

205887  ||  PR610 (hypoxia-activated prodrug, pan-HER inhibitor)

205626  ||  Pracinostat (SB939) (HDAC inhibitor)

202320  ||  Pralatrexate (dihydrofolate reductase inhibitor)

205865  ||  PRI-724 (CBP/beta-catenin antagonist; Wnt signaling pathway inhibitor)

202332  ||  Prinomastat

202334  ||  PRLX-93936

205597  ||  PRT-062607

205598  ||  PRX-302 (protein drug)

205599  ||  PTC-299 (VEGF inhibitor)

205601  ||  PTI-188 (a radiolabeled murine anti-melanin antibody)

205678  ||  PU-H71 (Hsp90 inhibitor)

205602  ||  PV-10

205745  ||  PWT33597 (PI3K inhibitor)

202340  ||  PX-12

202350  ||  PX-478 (HIF-1alpha inhibitor)

202360  ||  PX-866 (PI3K inhibitor)

202370  ||  Pyroxamide

205866  ||  PZP115891

205603  ||  QBI-139 (protein drug)

202380  ||  Quarfloxin (CX-3543) (G-quadruplex-interactive agent)

202385  ||  Quinacrine (Mepacrine ; CBLC102)

202390  ||  Quinagolide (D2 receptor agonist)

201612  ||  Quisinostat (JNJ-26481585) (HDAC inhibitor)

200072  ||  Quizartinib (AC220) (FLT3 inhibitor)

202391  ||  R1530 (Mitosis-angiogenesis inhibitor)

202411  ||  R306465 (JNJ-16241199)( HDAC inhibitor)

205926  ||  R406 (Syk inhibitor)

202420  ||  R547

202422  ||  R763 (AS703569) (Aurora kinase inhibitor)

205990  ||  Radotinib (tyrosine kinase inhibitor)

202430  ||  RC3095

202432  ||  RDEA-436 (MEK inhibitor)

205991  ||  Rebimastat (BMS-275291) (MMP inhibitor)

202431  ||  Refametinib (RDEA119;  BAY86-9766) (MEK inhibitor)

202436  ||  Regorafenib (BAY 73-4506) (oral multi-kinase inhibitor)

202440  ||  Relacatib

205867  ||  Resiquimod (Toll-like receptor (TLR) agonist)

205787  ||  Resminostat (4SC-201) (HDAC inhibitor)

202701  ||  Resveratrol(RM1812 , SRT-501)

202450  ||  Retaspimycin (IPI504) (HSP90 inhibitor)

205609  ||  RG-7167 (MEK inhibitor)

205917  ||  RG7388  (MDM2 antagonist)

202460  ||  RH1

200860  ||  Ridaforolimus (Deforolimus)

202080  ||  Rigosertib（ON-01910 ) (PLK1 inhibitor)

202701  ||  RM1812 (resveratrol, SRT-501)

202412  ||  RO4929097 (R4733) (gamma-secretase/Notch signalling pathway inhibitor)

202462  ||  RO4987655 (MEK inhibitor)

202421  ||  RO5045337 ( RG7112, R7112) (MDM2 (human homolog of double minutes-2; HDM2) antagonist)

205788  ||  RO5126766 (Raf/MEK dual kinase inhibitor)

205869  ||  RO518426 (V600E BRAF Blocker)

205611  ||  RO5212054 (PLX3603, RG-7256) (BRAF(V600E) kinase inhibitor)

205789  ||  RO5503781 (MDM2 antagonist)

202470  ||  Rolapitant (NK1 receptor antagonist)

202490  ||  Ropidoxuridine

202500  ||  Roquinimex (immunostimulant)

202510  ||  Rosabulin (STA-5312) (microtubule inhibitor)

202514  ||  Rostaporfin (PDT photosensitizer)

205870  ||  RRX-001 (radiosensitizer)

202540  ||  Rubitecan

200124  ||  Rucaparib (PF-01367338, AG-14699) (PARP1 inhibitor)

201512  ||  Ruxolitinib (INC-424;  INCB-18424) (JAK1 inhibitor)

202541  ||  S31-201

205992  ||  S-3304 (MMP inhibitor)

205767  ||  Sabarubicin (DNA intercalator)

203210  ||  Sagopilone (ZK epothilone)

202551  ||  Salirasib

202560  ||  Sapacitabine

205619  ||  SAR103168

205889  ||  SAR125844 (MEK inhibitor)

205623  ||  SAR3419

205624  ||  SAR411298 (FAAH inhibitor. Cancer pain)

200410  ||  Saracatinib (AZD-0530) (Src and Abl inhibitor)

200411  ||  Sardomozide ( SAMDC inhibitor)

201572  ||  Saridegib (IPI-926)  (Hedgehog pathway inhibitor)

202570  ||  Satraplatin 

205791  ||  SB-1518 (JAK2 inhibitor)

205790  ||  SB-743921 (KSP inhibitor)

205792  ||  SCH900353

202573  ||  SCH900776 (Chk1 inhibitor)

202580  ||  Seliciclib (CDK inhibitor)

200300  ||  Selumetinib (AZD-6244) (MEK 1/2 inhibitor)

202590  ||  Semapimod

205994  ||  Semaxanib (VEGFR2 inhibitor)

202600  ||  Seocalcitol (CB1089)

203190  ||  Sepantronium (YM-155) (Survivin inhibitor)

201614  ||  Serdemetan (JNJ-26854165)

202601  ||  SF1126

205629  ||  SGI-110 (DNMT inhibitor)

205710  ||  SGI-1776 (pan-Pim protein kinase inhibitor)

205630  ||  SGN-75 (anti-CD70 monoclonal antibody)

205715  ||  SGX-523 (Met Inhibitor)

205918  ||  SGX201 (active corticosteroid)

205871  ||  SHP-141 (HDAC inhibitor)

200274  ||  Silatecan (AR-67; DB-67) (topoisomerase I inhibitor; camptotecin derivative)

202610  ||  Silibinin ( extract of the milk thistle seeds; mixture of flavonolignans)

200843  ||  Silmitasertib (CX-4945) (CK2 inhibitor)

202620  ||  Simotaxel

205937  ||  Simotinib

200020  ||  Sivifene

200540  ||  SJG-136 (BN2629, SG2000) (DNA replication inhibitor)

202630  ||  SN-2310 (SN-38 conjugate with VE;  topoisomerase I inhibitor)

202640  ||  SNS-032 (BMS-387032) (CDK inhibitor)

202641  ||  SNS-314 (Aurora kinase inhibitor)

205736  ||  SNX-2112 (HSP90 inhibitor)

202651  ||  SNX-5422 (PF-4929113)

202660  ||  Soblidotin (tubulin polymerization inhibitor)

205627  ||  Sonoflora 1 ( SF1) (PDT photosensitizer)

205809  ||  Sotrastaurin (AEB071) (PCK inhibitor)

205872  ||  SPI-1005 (ebselen-containing oral capsule)

202680  ||  SPI-1620

202690  ||  Squalamine

205672  ||  SR13668 (Akt inhibitor)

206027  ||  SR4554 (bioreductive drug)

202700  ||  SR-31747 (Peripheral sigma receptor antagonist)

202702  ||  SSR97225

202715  ||  STA-1474 (Prodrug of ganetespib) (HSP90 inhibitor)

202708  ||  Stannsoporfin (heme oxygenase inhibitor)

202710  ||  SU14813

205633  ||  Sufentanil (ARX-02)

202713  ||  Sulforaphane (natural antioxidant)

205995  ||  Sulofenur (sulfonylurea)

205873  ||  SYP-0704A

205996  ||  T900607 (microtuble inhibitor)

205997  ||  Tacedinaline (HDAC inhibitor)

202045  ||  TAE684 (NVP-TAE684) (ALK Inhibitor)

202721  ||  TAK-285 (HER2/EGFR dual kinase inhibitor)

205919  ||  TAK-385 (GnRH receptor antagonist)

205635  ||  TAK-441 (Hedghog inhibitor)

205636  ||  TAK-448

202722  ||  TAK-593 (VEGFR/PDGFR dual kinase inhibitor)

202723  ||  TAK-683

205638  ||  TAK-733 (MEK inhibitor)

202725  ||  TAK-901 (Aurora B kinase inhibitor )

205639  ||  TAK-960 (PLK1 inhibitor)

202730  ||  Talabostat

202740  ||  Talampanel (AMPA-receptor antagonist)

202750  ||  Talaporfin sodium (PDT photosensitizer)

205998  ||  Talmapimod (MAKP inhibitor)

202770  ||  Talotrexin Ammonium

202760  ||  Taltobulin (tubulin inhibitor)

202780  ||  Tamibarotene (retinoic acid receptor (RAR) alpha/beta agonist)

202790  ||  Tandutinib (MLN0518) (tyrosine kinase inhibitor)

202953  ||  Tanomastat (matrix metalloprotease inhibitor)

100803  ||  Tapentadol

202810  ||  Tarenflurbil ((NSAID drug, enantiomer of flurbiprofen)

202820  ||  Tariquidar (p-glycoprotein inhibitor)

205641  ||  TAS-102

202834  ||  TAS-103 (BMS-247615)

202840  ||  TAS-108 (estrogenic receptor alpha (ERa) inhibitor)

202841  ||  TAS-109 (DNA polymerase inhibitor)

202850  ||  Tasidotin

202851  ||  Tasisulam (LY573636)

202852  ||  Tasquinimod (ABR-215050) (angiogenic inhibitor)

206001  ||  TCD-717 (CHKA inhibitor)

202860  ||  Teglarinad chloride (GMX-1777)

200680  ||  Telapristone (CDB-4124) (progesterone receptor modulator)

202950  ||  Telatinib ( Tanespimycin) (Hsp90 inhibitor)

206002  ||  Teloxantrone (topoisomerase II inhibitor)

202865  ||  Temoporfin (PDT photosensitizer)

202870  ||  Temsirolimus

202880  ||  Terameprocol (transcriptional inhibitor)

205875  ||  Teriflunomide (A77 1726; HMR1726) (Dihydrorotate dehydrogenase inhibitor; immunomodulatory drug)

202881  ||  Tesetaxel (DJ-927)

202890  ||  Tesmilifene

202900  ||  Tetrandrine

206004  ||   Tezacitabine (ribonucleotide reductase inhibitor)

205793  ||  TG-0054 (CXCR4 antagonist)

205642  ||  TG02 (multi-kinase inhibitor of CDKs, JAK2 and FLT3)

202892  ||  TG100-115 (PI3K inhibitor)

202893  ||  TG101348 ( JAK2 inhibitor)

205938  ||  TGR-1202 (PI3K delta inhibitor)

202895  ||  TGX-221 (PI3K inhibitor)

202901  ||  TH-302 (hypoxia-activated prodrug)

205643  ||  TH-9402

205644  ||  Thiarabine

202902  ||  Thymalfasin

201955  ||  Thymectacin (NB-1011).

206005  ||  Tiazofurin (IMPDH inhibitor)

202921  ||  Tigapotide

202926  ||  Timcodar (VX-853)

206006  ||  Timonacic

202930  ||  Tipifarnib (farnesyl transferase inhibitor)

206037  ||  Tipiracil (antimetabolite drug)

202940  ||  Tirapazamine (hypoxia toic agent)

200283  ||  Tivantinib (ARQ-197)  (c-Met inhibitor)

202955  ||  Tivozanib (AV-951) (VEGFR inhibitor)

202960  ||  TL-310 (a taxane)

205645  ||  TL32711 (Smac mimetic)

206007  ||  TLN-232 (pyruvate kinase inhibitor)

205738  ||  Toceranib (SU11654) (Hsp90 inhibitor)

200811  ||  Tofacitinib (CP-690550) (JAK inhibitor)

100880  ||  Toremifene

205648  ||  Tosedostat

202963  ||  Totrombopag

201900  ||  Tozasertib (MK-0457;  VX-680)  (Aurora inhibitor)

206003  ||  TPCS2a (Tetraphenyl chlorin disulfonate) (PDT photosensitizer)

202964  ||  TPI-287 (ARC-100)

202970  ||  Trabectedin

201458  ||  Trametinib (GSK-1120212, JTP-74057) (MEK 1/2 inhibitor)

205881  ||  Trastuzumab emtansine (trastuzumab (Herceptin) linked to the cytotoxin mertansine (DM1))

205652  ||  Treosulfan

202980  ||  Tretazicar (DNA alkylating agent)

203000  ||  Triapine (ribonucleotide reductase inhibitor)

203010  ||  Triciribine (VQD-002) (Akt inhibitor)

206038  ||  Trifluridine (antimetabolite drug)

203020  ||  Trilostane

206009  ||  TriN2755 (DNA cross linking agent)

205781  ||  Triphendiol

206010  ||  Trofosfamide (DNA cross linking agent)

203030  ||  Troxacitabine

203040  ||  TSU-68

206011  ||  TTP607 (Aurora kinase inhibitor)

203055  ||  Tubacin (HDAC6 inhibitor)

205939  ||  TW-37 (Bcl-2 inhibitor)

205655  ||  TXA127 (heptapeptide COX-2 inhibitor)

205931  ||  Tyroserleutide 

203070  ||  Ukrain

203071  ||  UNBS-5162

203160  ||  Upamostat (Mesupron, WX-671) (serine protease inhibitor)